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Replicase polyprotein 1ab inhibitor

Reticulon-4 inhibitor

Retinoic acid receptor agonist

Retinoic acid receptor alpha agonist

Retinoic acid receptor gamma agonist

Retinoid isomerohydrolase inhibitor

Retinoid receptor agonist

Retinoid X receptor agonist

Reverse transcriptase inhibitor

Rho-associated protein kinase inhibitor

Ribonucleoside-diphosphate reductase RR1 inhibitor

Ribosomal protein S6 kinase (P70S6K) inhibitor

Rivaroxaban sequestering agent

RNA-directed RNA polymerase L inhibitor

RNA disrupting agent

RNA inhibitor

Sclerostin inhibitor

Secretin receptor agonist

Selectin E antagonist

Serine-protein kinase ATR inhibitor

Serine/threonine-protein kinase AKT inhibitor

Serine/threonine-protein kinase Aurora-A inhibitor

Serine/threonine-protein kinase Aurora-B inhibitor

Serine/threonine-protein kinase Aurora inhibitor

Serine/threonine-protein kinase B-raf inhibitor

Serine/threonine-protein kinase Chk1 inhibitor

Serine/threonine-protein kinase Chk2 inhibitor

Serine/threonine-protein kinase mTOR inhibitor

Serine/threonine-protein kinase PIM inhibitor

Serine/threonine-protein kinase PLK1 inhibitor

Serine/threonine-protein kinase PLK4 inhibitor

Serine/threonine-protein kinase RAF inhibitor

Serine/threonine-protein kinase receptor R3 inhibitor

Serotonin 1a (5-HT1a) receptor agonist

Serotonin 1a (5-HT1a) receptor antagonist