Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Neoplasm Metastasis; Neuroendocrine Tumors
Unknown
Small molecule
Approved
Unknown
Unknown
Asthma; Hypersensitivity; Multiple Sclerosis; Rhinitis, Allergic, Seasonal; Chronic Urticaria; Inflammation; Lymphoma, Non-Hodgkin; Osteoarthritis, Knee; Pterygium
Unknown
Small molecule
Approved
OTHER
ORAL
Bacterial Infections
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
OTHER
INJECTION; ORAL
Carcinoma, Non-Small-Cell Lung; Depressive Disorder; Depressive Disorder, Major; Hypertension, Pulmonary; Leukemia, Myeloid, Acute; Lung Neoplasms; Prostatic Neoplasms; Altitude Sickness; Apnea; Hernias, Diaphragmatic, Congenital; Kidney Diseases; Leukemia; Pseudohypoparathyroidism; Renal Insufficiency, Chronic; Severe Acute Respiratory Syndrome; Virus Diseases; Pulmonary Disease, Chronic Obstructive; Respiratory Insufficiency; Asthma; Bronchitis, Chronic; Lung Diseases, Obstructive
Adenosine receptor antagonist
Small molecule
Approved
OTHER
INJECTION; ORAL; RECTAL
Altitude Sickness; Hypertension, Pulmonary; Premature Birth; Urinary Bladder Neoplasms; Heart Arrest; Acute Kidney Injury; Headache; Asthma; Lung Diseases, Obstructive
Adenosine receptor antagonist
Small molecule
Approved
OTHER
ORAL
Alopecia Areata; Bone Diseases, Metabolic; Colitis, Ulcerative; Colorectal Neoplasms; Diabetes, Gestational; Diabetes Mellitus, Type 2; Infertility; Inflammatory Bowel Diseases; Lung Neoplasms; Mood Disorders; Neoplasms; Penile Induration; Premature Birth; Sarcopenia; Anemia, Sickle Cell; Blood Coagulation Disorders; Crohn Disease; Death, Sudden, Cardiac; Diabetes Mellitus; Diabetic Neuropathies; Disseminated Intravascular Coagulation; Endometrial Neoplasms; Heart Failure; Hepatitis C; HIV Infections; Insulin Resistance; Latent Autoimmune Diabetes in Adults; Lupus Erythematosus, Cutaneous; Malnutrition; Migraine Disorders; Neuralgia; Optic Neuritis; Osteogenesis Imperfecta; Polycystic Ovary Syndrome; Prostatic Neoplasms; Restless Legs Syndrome; Spinal Cord Injuries; Uterine Cervical Neoplasms; Alzheimer Disease; Asthma; Breast Neoplasms; Burns; Cardiovascular Diseases; Cluster Headache; Colonic Neoplasms; Coronary Disease; Diabetes Mellitus, Type 1; Femoral Neck Fractures; Hepatitis C, Chronic; Hip Fractures; Hypocalcemia; Leukemia; Lipid Metabolism Disorders; Lymphoma; Lymphoma, Non-Hodgkin; Melanoma; Menopause; Multiple Sclerosis; Myocardial Ischemia; Neonatal Sepsis; Non-alcoholic Fatty Liver Disease; Obesity; Osteoarthritis, Knee; Osteoporosis; Osteoporosis, Postmenopausal; Pain; Pregnancy; Prostatic Neoplasms, Castration-Resistant; Renal Insufficiency, Chronic; Severe Acute Respiratory Syndrome; Tuberculosis; Tuberculosis, Pulmonary; Vitamin D Deficiency; Hypoparathyroidism; Hypophosphatemia, Familial; Rickets, Hypophosphatemic
Vitamin D receptor agonist
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Burns; Toxoplasmosis, Cerebral; Chorioretinitis; Toxoplasmosis, Congenital; Bacterial Infections; Malaria
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
Unknown
Unknown
Scoliosis; Ischemic Stroke; Sciatica; Pain
Unknown
Small molecule
Approved
CANCER; MUSCULOSKELETAL; OTHER; PREGNANCY AND GYNECOLOGY
INJECTION; ORAL; TOPICAL; VAGINAL
Memory; Reperfusion Injury; Brain Injuries; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Shock; Urinary Bladder, Overactive; Alzheimer Disease; Angina, Unstable; Anorexia Nervosa; Bone Diseases; Bone Diseases, Metabolic; Cardiovascular Diseases; Colonic Neoplasms; Coronary Disease; Cystitis, Interstitial; Diabetes Mellitus; Endometrial Neoplasms; Heart Diseases; Hot Flashes; Hypercholesterolemia; Hypertension; Lupus Erythematosus, Systemic; Memory Disorders; Myocardial Infarction; Myocardial Ischemia; Stroke; Thrombosis; Turner Syndrome; Atrophic Vaginitis; Atrophy; Breast Neoplasms; Dyspareunia; Hypogonadism; Menopause; Osteoporosis; Osteoporosis, Postmenopausal; Primary Ovarian Insufficiency
Estrogen receptor agonist
Small molecule
Approved
OTHER
ORAL
Digestive System Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Social Behavior; Amphetamine-Related Disorders; Obsessive-Compulsive Disorder; Attention Deficit Disorder with Hyperactivity
Unknown
Small molecule
Approved
OTHER
ORAL
Thrombosis
Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Acne Vulgaris; Conjunctivitis; Eye Infections; Infections
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
Unknown
Unknown
Bacterial Infections
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
TOPICAL
Osteomyelitis; Amyotrophic Lateral Sclerosis; Eye Infections; Leishmaniasis; Trypanosomiasis
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
alpha 1-Antitrypsin Deficiency; Crohn Disease; Depressive Disorder, Major; Dermatitis, Atopic; Fibrosis; Glycogen Storage Disease Type II; Hyperuricemia; Immune System Diseases; Lung Neoplasms; Mesothelioma; Purpura, Thrombocytopenic, Idiopathic; Alcoholism; Autistic Disorder; Breast Carcinoma In Situ; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Cocaine-Related Disorders; Endometrial Neoplasms; Graft vs Host Disease; Hepatitis B, Chronic; Immunoglobulin G4-Related Disease; Leukemia, Hairy Cell; Leukemia, Mast-Cell; Leukemia, Myeloid, Acute; Leukemia, T-Cell; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Myelodysplastic Syndromes; Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms, Castration-Resistant; Restless Legs Syndrome; Stomach Neoplasms; Stomatitis, Aphthous; Anxiety; Chronic Urticaria; Cough; Dementia; Depressive Disorder; Inflammation; Kidney Diseases; Lupus Erythematosus, Systemic; Lupus Nephritis; Migraine Disorders; Multiple Myeloma; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Pain; Rhinitis; Schizophrenia; Stomatitis; Urticaria; Hypersensitivity; Pruritus
Unknown
Small molecule
Approved
OTHER
INJECTION
Unknown
Heavy metals chelating agent
Small molecule
Approved
OTHER
ORAL
Epilepsy
Voltage-gated T-type calcium channel blocker
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Buruli Ulcer; Mycobacterium avium-intracellulare Infection; Plague; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Epilepsy
Sodium channel alpha subunit blocker
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Migraine with Aura; Migraine without Aura; Migraine Disorders
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Hemorrhage
Dopamine D1 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Hepatitis C; Premature Birth; Neonatal Abstinence Syndrome; Peripheral Nervous System Diseases; Restless Legs Syndrome; Cancer Pain; Chronic Pain; Cocaine-Related Disorders; Heroin Dependence; HIV Infections; Neoplasms; Neuralgia; Neuralgia, Postherpetic; Opioid-Related Disorders; Renal Insufficiency, Chronic; Scoliosis; Pain; Substance-Related Disorders
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Carcinoma, Squamous Cell; Neoplasms; Osteomyelitis; Stomach Neoplasms; Syphilis; Bacteremia; Infections; Pneumonia
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
VAGINAL
Unknown
Estrogen receptor alpha agonist
Small molecule
Approved
OTHER
ORAL
Ischemic Stroke; Graves Disease; Graves Ophthalmopathy; Thyrotoxicosis; Hyperthyroidism; Thyroid Diseases
Thyroid peroxidase inhibitor
Small molecule
Approved
Unknown
Unknown
Diabetes Mellitus, Type 2; Eosinophilic Esophagitis; Pancreatic Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Hypersensitivity
Unknown