| Synonyms: | |
| Status: | Phase 1 |
| Entry Type: | Small molecule |
| Molecule Category: | UNKNOWN |
| UNII: | E4768ZY6GM |
Physicochemical Descriptors
| Property Name | Value |
|---|---|
| Molecular Formula | C4H5AuO4S |
| Molecular Weight | 346.11 |
| AlogP | None |
| Hydrogen Bond Acceptor | None |
| Hydrogen Bond Donor | None |
| Number of Rotational Bond | None |
| Polar Surface Area | None |
| Molecular species | None |
| Aromatic Rings | None |
| Heavy Atoms | None |
Pharmacology
| Targets | EC50(nM) | IC50(nM) | Kd(nM) | Ki(nM) | Inhibition(%) | |
|---|---|---|---|---|---|---|
|
Enzyme
Kinase
Protein Kinase
TK protein kinase group
Tyrosine protein kinase EGFR family
|
- | 2379 | - | - | - | |
|
Enzyme
Kinase
Protein Kinase
TK protein kinase group
Tyrosine protein kinase Src family
|
- | 811 | - | - | - | |
|
Membrane receptor
Family A G protein-coupled receptor
Small molecule receptor (family A GPCR)
Nucleotide-like receptor (family A GPCR)
Adenosine receptor
|
- | 1492 | - | 843 | - |
Indications
| Mesh Heading | Maximum Phase | Mesh ID | Reference |
|---|---|---|---|
| Lung Neoplasms | 1 | D008175 | ClinicalTrials |
Cross References
| Resources | Reference |
|---|---|
| CAS NUMBER | 12244-57-4 |
| ChEBI | 38722 |
| ChEMBL | CHEMBL306043 |
| FDA SRS | E4768ZY6GM |
| PubChem | 422786 |
| SureChEMBL | SCHEMBL17874 |
CONTENTS