| Synonyms: | |
| Status: | Phase 2 |
| Entry Type: | Small molecule |
| Molecule Category: | UNKNOWN |
| UNII: | 63J9EQ81YC |
Physicochemical Descriptors
| Property Name | Value |
|---|---|
| Molecular Formula | C22H25N3O3 |
| Molecular Weight | 379.46 |
| AlogP | 3.6 |
| Hydrogen Bond Acceptor | 5.0 |
| Hydrogen Bond Donor | 1.0 |
| Number of Rotational Bond | 3.0 |
| Polar Surface Area | 65.37 |
| Molecular species | None |
| Aromatic Rings | 2.0 |
| Heavy Atoms | 28.0 |
Pharmacology
| Action | Mechanism of Action | Reference |
|---|---|---|
| ANTAGONIST | Histamine H1 receptor antagonist |
Indications
| Mesh Heading | Maximum Phase | Mesh ID | Reference |
|---|---|---|---|
| Sleep Initiation and Maintenance Disorders | 2 | D007319 | ClinicalTrials |
| Sleep Wake Disorders | 1 | D012893 | ClinicalTrials |
Cross References
| Resources | Reference |
|---|---|
| ChEMBL | CHEMBL3545287 |
| FDA SRS | 63J9EQ81YC |
CONTENTS