| Targets | EC50(nM) | IC50(nM) | Kd(nM) | Ki(nM) | Inhibition(%) | |
|---|---|---|---|---|---|---|
|
Membrane receptor
Family B G protein-coupled receptor
Peptide receptor (family B GPCR)
Calcitonin-like receptor
Calcitonin gene-related peptide receptor
|
562.34 | - | - | - | - | |
|
Membrane receptor
Family B G protein-coupled receptor
Peptide receptor (family B GPCR)
Calcitonin-like receptor
Calcitonin receptor
|
0.01862 | - | - | - | - | |
|
Other membrane protein
|
0.01862 | - | - | - | - | |
|
Unclassified protein
|
0.04677 | - | - | - | - |
| Mesh Heading | Maximum Phase | Mesh ID | Reference |
|---|---|---|---|
| Obesity | 1 | D009765 | ClinicalTrials |
| Resources | Reference |
|---|---|
| ChEMBL | CHEMBL4802169 |