Display Options:
Total: 6532
Small molecule
Approved
OTHER
TOPICAL
Psoriasis; Breast Neoplasms; Dermatitis, Atopic; Hemorrhoids; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Neoplasms; Common Cold; Conjunctivitis, Allergic; Influenza, Human; Eye Manifestations; Nasal Obstruction
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Osteomyelitis; Rhinoscleroma; Arthritis, Rheumatoid; Carcinoma, Non-Small-Cell Lung; Constipation; Coronary Disease; Diabetes Mellitus; Diabetes Mellitus, Type 2; Endometriosis; Essential Hypertension; Hepatitis B, Chronic; HIV Infections; Hodgkin Disease; Hypertension, Pulmonary; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma; Lymphoma, Non-Hodgkin; Melanoma; Mycoses; Nausea; Neoplasms; Non-alcoholic Fatty Liver Disease; Parkinson Disease; Renal Insufficiency; Renal Insufficiency, Chronic; Respiratory Syncytial Virus Infections; Sepsis; Thrombosis; Acquired Immunodeficiency Syndrome; Cystic Fibrosis; Meningitis; Multiple Sclerosis; Mycobacterium avium-intracellulare Infection; Onchocerciasis; Sarcoidosis; Alzheimer Disease; Arthritis, Reactive; Diarrhea; Endocarditis; Enterocolitis, Pseudomembranous; Infections; Leprosy; Multiple System Atrophy; Tuberculosis; Tuberculosis, Pulmonary
Bacterial DNA-directed RNA polymerase inhibitor
Small molecule
Approved
OTHER
ORAL
Carcinoma in Situ; Dementia; Head and Neck Neoplasms; HIV Wasting Syndrome; Pulmonary Disease, Chronic Obstructive; Uterine Neoplasms; Breast Neoplasms; Endometrial Hyperplasia; Endometrial Neoplasms; Hot Flashes; Liver Neoplasms; Acquired Immunodeficiency Syndrome; Anorexia; Cachexia; Neoplasms; Primary Immunodeficiency Diseases
Progesterone receptor agonist
Small molecule
Approved
OTHER
ORAL
Anxiety; Anxiety Disorders; Seizures
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
OTHER
ORAL
Unknown
Androgen Receptor agonist
Small molecule
Approved
DERMATOLOGY; OTHER
TOPICAL
Dermatitis, Atopic; Eye Diseases; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INTRAOCULAR
Presbyopia; Cataract; Glaucoma; Miosis
Muscarinic acetylcholine receptor M3 agonist
Small molecule
Approved
OTHER
OPHTHALMIC; TOPICAL
Corneal Opacity; Dry Eye Syndromes; Acne Vulgaris; Eye Diseases; Hemorrhoids; Inflammation
Glucocorticoid receptor agonist
Small molecule
Approved
CARDIOVASCULAR; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
BUCCAL; IMPLANTATION; INJECTION; NASAL; TRANSDERMAL
Cerebral Arterial Diseases; Dyspareunia; Insulin Resistance; Polycystic Ovary Syndrome; Aging; Kallmann Syndrome; Penile Induration; Acquired Immunodeficiency Syndrome; Anorexia Nervosa; Dwarfism; Heart Failure; Hereditary Breast and Ovarian Cancer Syndrome; Menopause; Multiple Sclerosis; Muscular Diseases; Obesity; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sarcopenia; Spinal Cord Injuries; Testicular Neoplasms; Coronary Disease; Disorders of Sex Development; Erectile Dysfunction; Hip Fractures; Infertility; Metabolic Syndrome; Neoplasms; Renal Insufficiency, Chronic; Sexual Dysfunction, Physiological; Hypogonadism; Klinefelter Syndrome; Orchitis
Androgen Receptor agonist
Small molecule
Approved
OTHER
INJECTION
Unknown
Muscle-type nicotinic acetylcholine receptor antagonist
Small molecule
Approved
OTHER
INJECTION
Psoriasis; Psychotic Disorders
Dopamine D2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
EMERGENCY MEDICINE; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
INJECTION
Neuralgia; Aortic Coarctation; Brain Neoplasms; HIV Infections; Prostatic Neoplasms, Castration-Resistant; Sinusitis; Vasospasm, Intracranial; Abdominal Pain; Appendicitis; Blepharoptosis; Blood Coagulation Disorders; Cleft Palate; Dupuytren Contracture; Fasciitis, Plantar; Femoral Neck Fractures; Headache; Hemorrhage; Hernia, Umbilical; Hip Fractures; Hypospadias; Hypotension; Lacrimal Apparatus Diseases; Low Back Pain; Lung Neoplasms; Mucositis; Osteoarthritis, Hip; Osteoarthritis, Knee; Pregnancy; Pulpitis; Rib Fractures; Rotator Cuff Injuries; Sarcoma; Shoulder Pain; Spinal Stenosis; Ankle Fractures; Breast Neoplasms; Breech Presentation; Carcinoma, Non-Small-Cell Lung; Chronic Pain; Cough; Fractures, Bone; Genital Neoplasms, Female; Hallux Valgus; Hemorrhoids; Hernia, Inguinal; Ileus; Liver Diseases; Migraine Disorders; Neoplasms; Osteoarthritis; Pancreatic Neoplasms; Pancreatitis, Chronic; Peritoneal Neoplasms; Postoperative Complications; Postoperative Nausea and Vomiting; Radiculopathy; Toothache; Urethral Stricture; Wounds and Injuries; Hernia; Pain
Sodium channel protein type IV alpha subunit blocker
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Prostatic Neoplasms, Castration-Resistant; Dental Caries; Gingivitis; Sensitivity and Specificity
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Postoperative Nausea and Vomiting; Vertigo; Vomiting
Histamine H1 receptor antagonist
Small molecule
Approved
OTHER
INHALATION
Unknown
GABA-A receptor; anion channel positive modulator
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Renal Insufficiency, Chronic; Cardiovascular Diseases; Heart Failure; Hypertension; Toxemia
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
Unknown
Unknown
Liver Neoplasms; Seminoma; Testicular Neoplasms; Neoplasms
Unknown
Small molecule
Unknown
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Coronary Disease; HIV Infections; Inflammation; Ischemia; Anemia; Anemia, Sickle Cell; Diabetes Mellitus, Type 2; Glaucoma
Unknown
Small molecule
Approved
OTHER
BUCCAL; ORAL; SUBLINGUAL
Menopause; Breast Neoplasms; Hypogonadism; Orchitis
Androgen Receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL; VAGINAL
Prostatic Neoplasms, Castration-Resistant; Neoplasms
Estrogen receptor alpha agonist
Small molecule
Approved
Unknown
Unknown
Obesity; Melanoma; Fractures, Bone; Arrhythmias, Cardiac; Bacteremia; Cellulitis; Gram-Positive Bacterial Infections; Infections; Laryngeal Neoplasms; Osteomyelitis; Prostatic Neoplasms, Castration-Resistant; Skin Diseases; Staphylococcal Infections; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Hypersensitivity; Pruritus
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Depressive Disorder; Diabetes Mellitus, Type 2; Obesity; Adenoma, Islet Cell; Hyperinsulinism; Hypertension; Hypoglycemia
Potassium channel, inwardly rectifying, subfamily J, member 11 opener
Small molecule
Unknown
Unknown
Unknown
Substance-Related Disorders; Asthma
Beta-2 adrenergic receptor agonist
Small molecule
Approved
OTHER
ORAL
Kidney Diseases; Graves Disease; Hyperlipoproteinemia Type II; Lipid Metabolism Disorders; Multiple Sclerosis; Myocardial Infarction; Myocardial Ischemia; Hypercholesterolemia; Hypothyroidism; Nephrotic Syndrome
Bile acids sequestering agent
Small molecule
Approved
Unknown
Unknown
Keratitis, Herpetic
Unknown
Small molecule
Approved
OTHER
ORAL
Rhinitis, Allergic, Seasonal
Histamine H1 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Infections; Burns
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Astrocytoma; Brain Neoplasms; Glioblastoma; Granulomatosis with Polyangiitis; Kidney Diseases; Leukemia, Biphenotypic, Acute; Neoplasms; Cystic Fibrosis; Dermatitis, Atopic; Diabetes Mellitus, Type 1; Eczema; Lymphoma, AIDS-Related; Abscess; HIV Infections; Idiopathic Pulmonary Fibrosis; Malaria; Measles; Pneumonia; Pyelonephritis; Sepsis; Staphylococcal Infections; Toxoplasmosis, Ocular; Tuberculosis; Bacterial Infections; Infections; Pneumonia, Pneumocystis; Urinary Tract Infections
Bacterial dihydropteroate synthase inhibitor