Display Options:
Total: 6532
Small molecule
Approved
OTHER
ORAL
Rhinitis, Allergic, Seasonal
Histamine H1 receptor antagonist
Small molecule
Unknown
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Hypersensitivity; Pruritus
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Depressive Disorder; Diabetes Mellitus, Type 2; Obesity; Adenoma, Islet Cell; Hyperinsulinism; Hypertension; Hypoglycemia
Potassium channel, inwardly rectifying, subfamily J, member 11 opener
Small molecule
Approved
Unknown
Unknown
Keratitis, Herpetic
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Adrenergic receptor alpha-1 agonist
Small molecule
Approved
OTHER
ORAL
Heart Diseases; Substance-Related Disorders; Brain Injuries; Status Epilepticus; Sleep Initiation and Maintenance Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Infections; Burns
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
Unknown
Unknown
Coronary Disease; HIV Infections; Inflammation; Ischemia; Anemia; Anemia, Sickle Cell; Diabetes Mellitus, Type 2; Glaucoma
Unknown
Small molecule
Approved
Unknown
Unknown
Depressive Disorder; Diabetes Mellitus; Cognitive Dysfunction; Heart Failure; Premature Birth; Hernias, Diaphragmatic, Congenital; Parkinson Disease; Shock; Shock, Septic; Cardiovascular Diseases
Unknown
Small molecule
Approved
IMMUNE SYSTEM; OTHER; PEDIATRICS
ORAL
Diarrhea; Inflammation; Osteomyelitis; Tooth Diseases; Astrocytoma; Brain Neoplasms; Central Serous Chorioretinopathy; Glioblastoma; Obesity; Obesity, Morbid; Postoperative Complications; Asthma; Bacteremia; Chlamydia Infections; Colitis, Ulcerative; Head and Neck Neoplasms; Lymphoma; Lymphoma, B-Cell, Marginal Zone; Mastitis; Periapical Periodontitis; Pneumonia, Bacterial; Pseudomyxoma Peritonei; Tuberculosis; Tuberculosis, Pulmonary; Vaginosis, Bacterial; Abscess; Bronchitis, Chronic; Cholecystitis; Communicable Diseases; Dyspepsia; Endocarditis; Enterobacteriaceae Infections; Fever; Gastritis; Helicobacter Infections; Hemorrhage; Hepatitis, Alcoholic; Low Back Pain; Lymphoma, Non-Hodgkin; Malaria; Neutropenia; Otitis Media, Suppurative; Periodontitis; Pyelonephritis; Severe Acute Respiratory Syndrome; Stomach Ulcer; Bacterial Infections; Duodenal Ulcer; Gonorrhea; Infections; Otitis Media; Pharyngitis; Pneumonia; Respiratory Tract Infections; Sinusitis; Soft Tissue Infections; Tonsillitis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
INTRAVENOUS; ORAL
Ankle Fractures; Alzheimer Disease; Hypotension, Orthostatic; Malaria; Muscular Dystrophy, Duchenne; Osteoarthritis, Knee; Premature Birth; Rhinitis, Allergic, Seasonal; Temporomandibular Joint Disorders; Brachial Plexus Neuritis; Bronchopulmonary Dysplasia; Cognitive Dysfunction; Depressive Disorder, Major; Diabetes Mellitus, Type 1; Emphysema; Enuresis; Epilepsies, Partial; Glioma; Granulomatous Disease, Chronic; Hemorrhage; Hypertension; Muscular Diseases; Pancreatitis; Periodontitis; Pre-Eclampsia; Retinopathy of Prematurity; Sinusitis; Spondylarthropathies; Spondylosis; Stomatitis, Aphthous; Sunburn; Tension-Type Headache; Tooth Diseases; Tuberculosis; Wounds and Injuries; Altitude Sickness; Breast Neoplasms; Burns; Causalgia; Cerebral Palsy; Chronic Pain; Fractures, Bone; HIV Infections; Hypospadias; Infections; Low Back Pain; Multiple Sclerosis; Neck Pain; Peptic Ulcer; Pulpitis; Respiratory Distress Syndrome; Shock, Septic; Sleep Apnea, Obstructive; Sprains and Strains; Vasculitis; Acute Pain; Arthralgia; Arthritis; Arthritis, Juvenile; Arthritis, Rheumatoid; Back Pain; Cardiovascular Diseases; Common Cold; Ductus Arteriosus, Patent; Dysmenorrhea; Fever; Headache; Influenza, Human; Migraine Disorders; Muscle Cramp; Myalgia; Osteoarthritis; Pain; Pharyngitis; Rheumatic Diseases; Toothache; Vaginitis
Cyclooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Gram-Positive Bacterial Infections; Mastitis; Enterobacteriaceae Infections; Staphylococcal Infections; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Bacterial Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
ORAL
Glioma; Hookworm Infections; Pruritus; Anemia; Colorectal Neoplasms; Necatoriasis; Helminthiasis
Tubulin inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Bile acids sequestering agent
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
TOPICAL
Lice Infestations; Ectoparasitic Infestations
GABA-A receptor negative allosteric modulator
Small molecule
Approved
Unknown
Unknown
Multiple Sclerosis; Fever; Tachycardia, Ventricular; Wounds and Injuries
Unknown
Small molecule
Approved
OTHER
INJECTION
Atrophic Vaginitis
Androgen Receptor agonist
Small molecule
Approved
OTHER
ORAL
Neoplasms; Prostatic Neoplasms, Castration-Resistant; Small Cell Lung Carcinoma; Carcinoma, Squamous Cell; Hypertension; Laryngeal Neoplasms; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Prostatic Neoplasms; Angina, Stable
Unknown
Small molecule
Approved
OTHER
INJECTION
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Hypersensitivity
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Carnitine O-palmitoyltransferase 1, muscle isoform inhibitor
Small molecule
Approved
Unknown
Unknown
Diabetic Cardiomyopathies; Heart Failure; Heart Failure, Diastolic; Cardiomyopathy, Hypertrophic; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Diabetes Mellitus, Type 1; Neuralgia; Asthma; Pulmonary Disease, Chronic Obstructive; Lung Diseases, Obstructive
Unknown
Small molecule
Approved
Unknown
Unknown
Bacterial Infections
Unknown
Small molecule
Unknown
Unknown
Unknown
Bacterial Infections
Unknown
Small molecule
Approved
IMMUNE SYSTEM; PREGNANCY AND GYNECOLOGY
BUCCAL; INJECTION
Intertrigo; Stomatitis; HIV Infections; Infections; Mycoses; Pruritus; Tinea; Tinea Pedis
Cytochrome P450 51 inhibitor
Small molecule
Approved
Unknown
Unknown
Diabetes Mellitus, Type 2; Diabetes Mellitus
Acyl coenzyme A:cholesterol acyltransferase 1 inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION
Unknown
Unknown
Small molecule
Approved
OTHER
OPHTHALMIC
Urinary Incontinence; Presbyopia; Glaucoma; Glaucoma, Angle-Closure; Glaucoma, Open-Angle; Miosis; Ocular Hypertension; Sjogren's Syndrome; Xerostomia
Muscarinic acetylcholine receptor M1 agonist