Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Unknown
Progesterone receptor agonist
Small molecule
Approved
OTHER
ORAL; TOPICAL
Adenoma; Hypospadias; Oral Ulcer; Bronchiolitis; Dermatitis, Atopic; Dry Eye Syndromes; Glaucoma; Hyaline Membrane Disease; Macular Edema; Melanoma; Neck Pain; Respiratory Distress Syndrome, Newborn; Retinal Vein Occlusion; Sciatica; Tachypnea; Carpal Tunnel Syndrome; Cough; Eczema; Gout; Hypersensitivity; Lichen Planus, Oral; Orbital Pseudotumor; Pharyngitis; Pregnancy; Premature Birth; Psoriasis; Respiratory Distress Syndrome; Rhinitis, Allergic, Seasonal; Eye Diseases; Hemorrhoids; Lung Diseases, Obstructive; Nasal Obstruction
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
ORAL
Chronic Pain; Endotoxemia; Hepatitis C, Chronic; Lymphoma; Neoplasms; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
OTHER
ORAL
Cocaine-Related Disorders; Tobacco Use Disorder; Depressive Disorder, Major; Cushing Syndrome; Depressive Disorder
Cytochrome P450 11B1, mitochondrial inhibitor
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Hernia, Inguinal; Hypersensitivity
Unknown
Small molecule
Approved
Unknown
Unknown
Depressive Disorder
Unknown
Small molecule
Approved
Unknown
Unknown
Migraine Disorders
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
Serotonin 1a (5-HT1a) receptor partial agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION; INTRAVESICAL; URETERAL
Unknown
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Candidiasis; Infections; Tinea; Tinea Capitis; Tinea Pedis
Tubulin inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Neoplasms
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Diabetes Mellitus, Type 1; Pre-Eclampsia; Hypertension
Adrenergic receptor alpha-2 agonist
Small molecule
Approved
Unknown
Unknown
Leukemia, Myeloid, Acute; Anxiety; Dementia; Depressive Disorder; Schizophrenia; Psychotic Disorders
D2-like dopamine receptor antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Myelodysplastic Syndromes
Androgen Receptor agonist
Small molecule
Approved
OTHER
ORAL
Unknown
Muscarinic acetylcholine receptor M1 antagonist
Small molecule
Approved
OTHER
INJECTION; ORAL; RECTAL
Landau-Kleffner Syndrome; Low Back Pain; Rotator Cuff Injuries; Wounds and Injuries; Dementia; Depressive Disorder; Epilepsy, Complex Partial; Pain; Schizophrenia; Seizures; Status Epilepticus; Vertigo; Anxiety; Anxiety Disorders; Cerebral Palsy; Epilepsy; Mental Disorders; Psychomotor Agitation; Stiff-Person Syndrome
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
DERMATOLOGY; IMMUNE SYSTEM; OTHER; PREGNANCY AND GYNECOLOGY
INJECTION; ORAL; TOPICAL; VAGINAL
Central Serous Chorioretinopathy; Cholangitis, Sclerosing; Osteomyelitis; Periapical Periodontitis; Pouchitis; Prostatic Neoplasms, Castration-Resistant; Appendicitis; Brain Diseases; Carcinoma, Non-Small-Cell Lung; Clostridium Infections; Colitis, Ulcerative; Giardiasis; Leukemia, Lymphocytic, Chronic, B-Cell; Lichen Planus, Oral; Malnutrition; Pancreatic Neoplasms; Periodontal Diseases; Pilonidal Sinus; Rectal Neoplasms; Tuberculosis; Tuberculosis, Multidrug-Resistant; Uterine Cervical Neoplasms; Abscess; Blepharitis; Candidiasis; Colorectal Neoplasms; Crohn Disease; Diarrhea; Enterocolitis, Pseudomembranous; Fecal Incontinence; Gingivitis; Helicobacter Infections; Hemorrhoids; Hidradenitis Suppurativa; HIV Infections; Lymphoma, Non-Hodgkin; Mycoses; Pain; Pelvic Inflammatory Disease; Periodontitis; Skin Diseases; Trichomonas Vaginitis; Vaginal Discharge; Vaginitis; Amebiasis; Bacterial Infections; Duodenal Ulcer; Infections; Intraabdominal Infections; Pneumonia; Rosacea; Sepsis; Trichomonas Infections; Uterine Cervicitis; Vaginosis, Bacterial
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Hypersensitivity; Hypotension, Orthostatic; Multiple System Atrophy; Cough; Inflammation; Respiratory Tract Infections; Rhinitis; Rhinitis, Allergic, Perennial; Rhinitis, Vasomotor; Common Cold; Nasal Obstruction; Rhinitis, Allergic, Seasonal
Unknown
Small molecule
Approved
OTHER
INTRAVITREAL; OTIC; TOPICAL
Glaucoma; Macular Degeneration; Retinal Diseases; Uveitis, Anterior; Uveitis, Intermediate; Uveitis, Posterior; Dermatitis, Atopic; Dermatitis, Seborrheic; Eye Diseases; Hemorrhoids; Infections; Macular Edema; Melanosis; Psoriasis; Skin Diseases; Uveitis
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Castleman Disease; Lymphoma, B-Cell; Lymphoma, Primary Effusion; Neoplasm Metastasis; Osteosarcoma; Sarcoma; Adrenal Cortex Neoplasms; Astrocytoma; Blast Crisis; Blastic Plasmacytoid Dendritic Cell Neoplasm; Burkitt Lymphoma; Glioblastoma; Hemangioma; Hematologic Neoplasms; Immunoblastic Lymphadenopathy; Leukemia, Biphenotypic, Acute; Lymphoma, Large-Cell, Anaplastic; Lymphoma, T-Cell; Purpura, Thrombocytopenic, Idiopathic; Rhabdomyosarcoma; Wilms Tumor; Brain Neoplasms; Central Nervous System Neoplasms; Choroid Plexus Neoplasms; Ependymoma; Ganglioneuroblastoma; Gestational Trophoblastic Disease; Glioma; Hepatoblastoma; Histiocytosis, Langerhans-Cell; HIV Infections; Hodgkin Disease; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Lymphoid; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Myeloid, Acute; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Medulloblastoma; Multiple Myeloma; Neuroblastoma; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Retinoblastoma; Rhabdomyosarcoma, Alveolar; Rhabdomyosarcoma, Embryonal; Sarcoma, Ewing; Small Cell Lung Carcinoma; Waldenstrom Macroglobulinemia; Neoplasms
Unknown
Small molecule
Approved
OTHER
ORAL
Rhinitis, Allergic, Seasonal
Histamine H1 receptor antagonist
Small molecule
Approved
OTHER
OPHTHALMIC
Leukemia; Eye Infections; Virus Diseases
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Cardiovascular Diseases
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
Unknown
Unknown
Hypersensitivity
Unknown
Small molecule
Approved
OTHER
INHALATION; INTRAVENOUS; ORAL
Aging; Altitude Sickness; Alzheimer Disease; Anosmia; beta-Thalassemia; Breast Neoplasms; Cardiomyopathy, Hypertrophic; Cystinosis; Depressive Disorder; Depressive Disorder, Major; Diabetes Mellitus, Type 2; Fibromyalgia; Gambling; Hearing Loss, Noise-Induced; HIV Infections; Irritable Bowel Syndrome; Lymphoma; Mitochondrial Diseases; Neuromuscular Diseases; Niemann-Pick Disease, Type C; Non-alcoholic Fatty Liver Disease; Pancreatitis; Persian Gulf Syndrome; Polycythemia Vera; Primary Myelofibrosis; Pseudomyxoma Peritonei; Purpura, Thrombotic Thrombocytopenic; Renal Insufficiency; Respiratory Distress Syndrome; Respiratory Tract Infections; Substance-Related Disorders; Thrombocythemia, Essential; Acute Lung Injury; Adrenoleukodystrophy; Alcohol Drinking; Alcoholism; Amphetamine-Related Disorders; Arrhythmias, Cardiac; Asperger Syndrome; Autistic Disorder; Bacteremia; Biliary Atresia; Bipolar Disorder; Brain Injuries; Bronchitis, Chronic; Child Development Disorders, Pervasive; Cocaine-Related Disorders; Cognitive Dysfunction; De Lange Syndrome; Dry Eye Syndromes; Epilepsy; Fuchs' Endothelial Dystrophy; Gaucher Disease; Hearing Loss; Hepatic Veno-Occlusive Disease; Homocystinuria; Huntington Disease; Ischemic Stroke; Kidney Diseases; Leiomyoma; Leukemia, Myeloid, Acute; Lupus Erythematosus, Systemic; Melanoma; Mental Disorders; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Muscular Diseases; Neuralgia; Neurofibromatosis 1; Obsessive-Compulsive Disorder; Parkinson Disease; Polycystic Ovary Syndrome; Premature Birth; Purpura, Thrombocytopenic, Idiopathic; Pyelonephritis; Rhabdomyolysis; Scleroderma, Diffuse; ST Elevation Myocardial Infarction; Stomatitis; Stress Disorders, Post-Traumatic; Stroke; Thrombocytopenia; Tobacco Use Disorder; Tourette Syndrome; Transposition of Great Vessels; Trichotillomania; Tuberculosis; Acute Kidney Injury; Anemia, Sickle Cell; Atrial Fibrillation; Bulimia Nervosa; Common Cold; Coronary Disease; Diabetic Foot; Graft vs Host Disease; Hematologic Diseases; Hepatitis, Alcoholic; Idiopathic Pulmonary Fibrosis; Infertility; Infertility, Female; Influenza, Human; Jaundice; Kidney Failure, Chronic; Liver Failure, Acute; Macular Degeneration; Marijuana Abuse; Mucositis; Myocardial Infarction; Psoriasis; Psychotic Disorders; Pulmonary Disease, Chronic Obstructive; Pulmonary Fibrosis; Renal Insufficiency, Chronic; Reperfusion Injury; Respiratory Tract Diseases; Retinitis Pigmentosa; Schizophrenia; Severe Acute Respiratory Syndrome; Sinusitis; Thrombosis; Chemical and Drug Induced Liver Injury; Cystic Fibrosis; Eye Diseases; Wounds and Injuries
Glutathione precursor
Small molecule
Approved
OTHER
ORAL
Atherosclerosis; Coronary Disease; Death, Sudden, Cardiac; Diabetes Mellitus, Type 2; Hypercholesterolemia; Cardiovascular Diseases; Edema; Heart Failure; Hyperaldosteronism; Hypertension; Liver Cirrhosis; Nephrotic Syndrome; Toxemia
Amiloride-sensitive sodium channel, ENaC blocker
Small molecule
Approved
OTHER
ORAL; TOPICAL; VAGINAL
Dental Caries; Kidney Diseases; Macular Degeneration; Bacteremia; Burns; Graft vs Host Disease; Pneumonia; Stomatitis, Denture; Candidiasis, Oral; HIV Infections; Leukemia; Lymphoma; Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Stomatitis; Tobacco Use Disorder; Vaginosis, Bacterial; Candidiasis; Infections
Ergosterol sequestering agent
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections; Multiple Sclerosis
Bacterial 70S ribosome inhibitor