Display Options:
Total: 6532
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Irritable Bowel Syndrome; Sleep Initiation and Maintenance Disorders; Anxiety; Dementia; Schizophrenia; Depressive Disorder; Pruritus
Unknown
Small molecule
Approved
OTHER
OPHTHALMIC
Unknown
Adrenergic receptor agonist
Small molecule
Approved
OTHER
OPHTHALMIC
Eye Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
INJECTION
Arthritis, Rheumatoid; Pain; Eye Diseases; Hemorrhoids; Lung Diseases, Obstructive; Nasal Obstruction; Osteoarthritis
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
INJECTION; ORAL
Puberty, Precocious
Cytochrome P450 19A1 inhibitor
Small molecule
Unknown
Unknown
Unknown
Astrocytoma; Glioblastoma; Lymphoma, AIDS-Related; Brain Neoplasms; Central Nervous System Neoplasms; Lymphoma
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION
Alopecia; Brain Neoplasms; Glioblastoma; Leukemia, Plasma Cell; Polycythemia Vera; Primary Myelofibrosis; Thrombocythemia, Essential; Blast Crisis; Burkitt Lymphoma; Central Nervous System Neoplasms; Hematologic Neoplasms; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Myelomonocytic, Juvenile; Lupus Erythematosus, Systemic; Lymphoma, AIDS-Related; Lymphoma, Large-Cell, Anaplastic; Lymphoma, T-Cell, Peripheral; Medulloblastoma; Meningitis, Aseptic; Multiple Sclerosis, Relapsing-Remitting; Myasthenia Gravis; Neuromyelitis Optica; Neutropenia; Opsoclonus-Myoclonus Syndrome; Ovarian Neoplasms; Polyradiculoneuropathy, Chronic Inflammatory Demyelinating; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Stiff-Person Syndrome; Urinary Bladder, Overactive; Anemia, Refractory; Anemia, Refractory, with Excess of Blasts; Breast Neoplasms; Graft vs Host Disease; Histiocytosis, Langerhans-Cell; Hodgkin Disease; Leukemia; Leukemia, Basophilic, Acute; Leukemia, Biphenotypic, Acute; Leukemia, Erythroblastic, Acute; Leukemia, Megakaryoblastic, Acute; Leukemia, Monocytic, Acute; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myelomonocytic, Acute; Leukemia, Myelomonocytic, Chronic; Leukemia, Promyelocytic, Acute; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Malaria; Melanoma; Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Renal Insufficiency, Chronic; Sarcoma, Myeloid; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Meningeal Carcinomatosis; Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Bacterial Infections
70S ribosome inhibitor
Small molecule
Approved
Unknown
Unknown
Osteomyelitis
Unknown
Small molecule
Approved
OTHER
INHALATION; ORAL
Brain Injuries; Amyotrophic Lateral Sclerosis; Asthma; Hypotension, Orthostatic; Tobacco Use Disorder; Tourette Syndrome; Albinism; Albinism, Oculocutaneous; Angelman Syndrome; Aphasia; Back Pain; Child Development Disorders, Pervasive; Cocaine-Related Disorders; Macular Degeneration; Pain; Retinitis Pigmentosa; Schizophrenia; Spinal Cord Injuries; Stress Disorders, Post-Traumatic; Amblyopia; Restless Legs Syndrome; Stroke; Parkinson Disease
Dopamine D3 receptor agonist
Small molecule
Approved
OTHER
ORAL
Unknown
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Sleep Initiation and Maintenance Disorders; Anxiety; Dementia; Depressive Disorder; Schizophrenia
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Unknown
Dopamine D2 receptor antagonist
Small molecule
Unknown
Unknown
Unknown
Pain; Postoperative Nausea and Vomiting; Psychotic Disorders
D2-like dopamine receptor antagonist
Small molecule
Approved
Unknown
Unknown
Polyuria; Urinary Incontinence
Unknown
Small molecule
Approved
OTHER
ORAL
Prostatic Neoplasms, Castration-Resistant; Adrenal Cortex Neoplasms; Carcinoma; Neoplasms
Cytochrome P450 11A1 inhibitor
Small molecule
Approved
OTHER
ORAL
Central Nervous System Neoplasms; Arthritis, Rheumatoid; Cystinuria; Hepatolenticular Degeneration; Inflammation; Rheumatic Diseases; Spondylitis
Copper chelating agent
Small molecule
Approved
OTHER
INJECTION
Sarcoma, Ewing; Neoplasms
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Hemorrhoids; Phobia, Social; Radius Fractures; Cognitive Dysfunction; Fatigue; Heart Arrest; Marijuana Abuse; Mental Disorders; Opioid-Related Disorders; Perceptual Disorders; Schizophrenia; Sepsis; Stroke; Substance-Related Disorders; Tobacco Use Disorder; Borderline Personality Disorder; Brain Injuries; Breast Neoplasms; Bronchial Spasm; Child Development Disorders, Pervasive; Cocaine-Related Disorders; Complex Regional Pain Syndromes; Coronavirus Infections; Depressive Disorder, Treatment-Resistant; Epilepsy; Fractures, Multiple; Heart Septal Defects, Ventricular; Hypertrophy; Ischemic Stroke; Lung Neoplasms; Obsessive-Compulsive Disorder; Paget Disease, Extramammary; Respiratory Distress Syndrome; Rett Syndrome; Severe Acute Respiratory Syndrome; Strabismus; Stress Disorders, Post-Traumatic; Subarachnoid Hemorrhage; Temporomandibular Joint Disorders; Alcoholism; Anemia, Sickle Cell; Bipolar Disorder; Chronic Pain; Delirium; Depression, Postpartum; Depressive Disorder; Depressive Disorder, Major; Fractures, Bone; Headache; Mucositis; Neoplasms; Neuralgia; Obesity, Morbid; Pain; Pharyngitis; Postoperative Complications; Renal Colic; Rib Fractures; Shock, Septic; Status Asthmaticus; Status Epilepticus; Suicidal Ideation; Wounds and Injuries
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Dermatitis, Atopic; Epidermolysis Bullosa Dystrophica; Muscular Dystrophy, Duchenne; Pneumonia, Ventilator-Associated; Chorioamnionitis; Cystic Fibrosis; Diabetic Foot; Folliculitis; Leishmaniasis; Leishmaniasis, Cutaneous; Meniere Disease; Neoplasms; Plague; Breast Neoplasms; Cat-Scratch Disease; Colonic Neoplasms; Eczema; Infections; Pain; Rectal Neoplasms; Sepsis; Bacterial Infections; Eye Infections
Unknown
Small molecule
Unknown
Unknown
Unknown
Psychotic Disorders
Unknown
Small molecule
Approved
Unknown
Unknown
Vaginitis; Sepsis; Periapical Periodontitis; Prediabetic State; Severe Acute Respiratory Syndrome; Breast Neoplasms; Candidiasis, Vulvovaginal; Chorioretinitis; Kidney Calculi; Malaria; Nasal Obstruction; Pain; Pneumonia, Pneumocystis; Skin Diseases; Staphylococcal Infections; Vaginosis, Bacterial; Acne Vulgaris; Bacterial Infections; Endometritis; Infections; Intraabdominal Infections; Osteomyelitis
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Neuroendocrine Tumors; Psoriasis; Melanoma; Tobacco Use Disorder
Unknown
Small molecule
Approved
OTHER
ORAL
Astrocytoma; Carcinoma, Hepatocellular; Colorectal Neoplasms; Gliosarcoma; Neoplasms; Oligodendroglioma; Intracranial Hypertension; Meningitis, Cryptococcal; Candidiasis; Infections; Meningitis
Thymidylate synthase inhibitor
Small molecule
Approved
OTHER
INJECTION; ORAL
Osteomyelitis; Rhinoscleroma; Arthritis, Rheumatoid; Carcinoma, Non-Small-Cell Lung; Constipation; Coronary Disease; Diabetes Mellitus; Diabetes Mellitus, Type 2; Endometriosis; Essential Hypertension; Hepatitis B, Chronic; HIV Infections; Hodgkin Disease; Hypertension, Pulmonary; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma; Lymphoma, Non-Hodgkin; Melanoma; Mycoses; Nausea; Neoplasms; Non-alcoholic Fatty Liver Disease; Parkinson Disease; Renal Insufficiency; Renal Insufficiency, Chronic; Respiratory Syncytial Virus Infections; Sepsis; Thrombosis; Acquired Immunodeficiency Syndrome; Cystic Fibrosis; Meningitis; Multiple Sclerosis; Mycobacterium avium-intracellulare Infection; Onchocerciasis; Sarcoidosis; Alzheimer Disease; Arthritis, Reactive; Diarrhea; Endocarditis; Enterocolitis, Pseudomembranous; Infections; Leprosy; Multiple System Atrophy; Tuberculosis; Tuberculosis, Pulmonary
Bacterial DNA-directed RNA polymerase inhibitor
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Alcoholism; Autistic Disorder; Brain Injuries; Carcinoma, Non-Small-Cell Lung; Cerebral Hemorrhage; Child Development Disorders, Pervasive; Cholangitis, Sclerosing; Fibromyalgia; Glioblastoma; Glioma; Hemorrhage; Memory Disorders; Periapical Periodontitis; Pneumonia; Retinal Vein Occlusion; Skin Diseases; Angelman Syndrome; Asthma; Atrial Fibrillation; Carotid Stenosis; Chronic Pain; Colorectal Neoplasms; Cystic Fibrosis; Depressive Disorder, Major; Esophageal Neoplasms; Fragile X Syndrome; Head and Neck Neoplasms; HIV Infections; Huntington Disease; Impetigo; Lung Neoplasms; Macular Degeneration; Multiple Myeloma; Multiple Sclerosis, Relapsing-Remitting; Neuralgia; Obsessive-Compulsive Disorder; Oropharyngeal Neoplasms; Pancreatic Neoplasms; Parkinson Disease; Retinal Detachment; Retinitis Pigmentosa; Stroke; Amyotrophic Lateral Sclerosis; Arthritis, Rheumatoid; Bipolar Disorder; Depressive Disorder; Depressive Disorder, Treatment-Resistant; Heroin Dependence; Hypertension; Idiopathic Pulmonary Fibrosis; Lichen Planus, Oral; Multiple Sclerosis; Neurobehavioral Manifestations; Peri-Implantitis; Periodontitis; Pneumothorax; Psychotic Disorders; Rosacea; Schizophrenia; Spinal Cord Injuries; Acne Vulgaris; Bacterial Infections; Infections
Unknown
Small molecule
Approved
OTHER
TOPICAL
Psoriasis; Breast Neoplasms; Dermatitis, Atopic; Hemorrhoids; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
DERMATOLOGY; OTHER
ORAL; TOPICAL
Hypercholesterolemia; Amyotrophic Lateral Sclerosis; Hematologic Neoplasms; Myelodysplastic-Myeloproliferative Diseases; Anemia; Anti-Neutrophil Cytoplasmic Antibody-Associated Vasculitis; Breast Neoplasms; Carcinoma, Adenoid Cystic; Cholangitis, Sclerosing; Emphysema; Keratosis, Actinic; Kidney Neoplasms; Lentigo; Lung Neoplasms; Lymphoma; Melanoma; Multiple Myeloma; Neuroblastoma; Pancreatic Neoplasms; Prostatic Neoplasms; Severe Acute Respiratory Syndrome; Small Cell Lung Carcinoma; Carcinoma, Basal Cell; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Leukemia; Leukemia, Myeloid, Acute; Myelodysplastic Syndromes; Myeloproliferative Disorders; Purpura, Thrombocytopenic, Idiopathic; Rosacea; Acne Vulgaris; Hyperpigmentation; Leukemia, Promyelocytic, Acute; Melanosis; Neoplasms
Retinoic acid receptor agonist
Small molecule
Approved
OTHER
ORAL
Carcinoma in Situ; Dementia; Head and Neck Neoplasms; HIV Wasting Syndrome; Pulmonary Disease, Chronic Obstructive; Uterine Neoplasms; Breast Neoplasms; Endometrial Hyperplasia; Endometrial Neoplasms; Hot Flashes; Liver Neoplasms; Acquired Immunodeficiency Syndrome; Anorexia; Cachexia; Neoplasms; Primary Immunodeficiency Diseases
Progesterone receptor agonist
Small molecule
Approved
Unknown
Unknown
Neoplasms; Common Cold; Conjunctivitis, Allergic; Influenza, Human; Eye Manifestations; Nasal Obstruction
Unknown
Small molecule
Approved
OTHER
ORAL
Pain
Mu opioid receptor agonist
Small molecule
Approved
Unknown
Unknown
Infections; Bacteremia; Gram-Positive Bacterial Infections; Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Unknown
Unknown
Unknown
Leukemia, Myeloid, Acute; Urinary Bladder, Overactive; Cellulitis; Dermatitis, Atopic; Eczema; Staphylococcal Infections; Urinary Tract Infections; Cystic Fibrosis; Nasal Obstruction; Skin Diseases; Urinary Bladder Neoplasms; Bacterial Infections; Infections; Otitis Media; Prostatitis; Respiratory Tract Infections; Sprains and Strains
Bacterial penicillin-binding protein inhibitor