Display Options:
Total: 6532
Small molecule
Approved
OTHER
INJECTION
Brain Neoplasms; Glioblastoma; Leukemia, Plasma Cell; Paraganglioma; Polycythemia Vera; Primary Myelofibrosis; Thrombocythemia, Essential; Blast Crisis; Blastic Plasmacytoid Dendritic Cell Neoplasm; Burkitt Lymphoma; Central Nervous System Neoplasms; Hematologic Neoplasms; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Myelomonocytic, Juvenile; Lupus Erythematosus, Systemic; Lymphoma, AIDS-Related; Lymphoma, Large-Cell, Anaplastic; Lymphoma, T-Cell, Peripheral; Medulloblastoma; Meningitis, Aseptic; Multiple Sclerosis, Relapsing-Remitting; Myasthenia Gravis; Neoplasms, Plasma Cell; Neuromyelitis Optica; Neutropenia; Opsoclonus-Myoclonus Syndrome; Ovarian Neoplasms; Polyradiculoneuropathy, Chronic Inflammatory Demyelinating; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Stiff-Person Syndrome; Anemia, Refractory; Anemia, Refractory, with Excess of Blasts; Breast Neoplasms; Graft vs Host Disease; Histiocytosis, Langerhans-Cell; Hodgkin Disease; Leukemia; Leukemia, Basophilic, Acute; Leukemia, Biphenotypic, Acute; Leukemia, Erythroblastic, Acute; Leukemia, Megakaryoblastic, Acute; Leukemia, Monocytic, Acute; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid; Leukemia, Myelomonocytic, Acute; Leukemia, Myelomonocytic, Chronic; Leukemia, Promyelocytic, Acute; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Malaria; Melanoma; Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Sarcoma, Myeloid; Thrombosis; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Meningeal Carcinomatosis; Meningeal Neoplasms; Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Glioblastoma; Central Nervous System Neoplasms; Hodgkin Disease; Lymphoma; Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Irritable Bowel Syndrome; Sleep Wake Disorders; Anxiety; Dementia; Schizophrenia; Urticaria; Depressive Disorder; Pruritus
Histamine H1 receptor antagonist
Small molecule
Approved
OTHER
ORAL
Unknown
Dopamine D2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Leishmaniasis; Leishmaniasis, Cutaneous; Leishmaniasis, Visceral
Unknown
Small molecule
Approved
Unknown
Unknown
Astrocytoma; Glioblastoma; Lymphoma, AIDS-Related; Brain Neoplasms; Central Nervous System Neoplasms; Lymphoma
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INJECTION
Arthritis, Rheumatoid; Joint Diseases; Pain; Osteoarthritis, Knee; Osteoarthritis
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Puberty, Precocious
Cytochrome P450 19A1 inhibitor
Small molecule
Approved
Unknown
Unknown
Dermatitis, Atopic; Epidermolysis Bullosa Dystrophica; Muscular Dystrophy, Duchenne; Osteomyelitis; Pneumonia, Ventilator-Associated; Chorioamnionitis; Cystic Fibrosis; Diabetic Foot; Folliculitis; Leishmaniasis; Leishmaniasis, Cutaneous; Meniere Disease; Neoplasms; Urinary Tract Infections; Breast Neoplasms; Cat-Scratch Disease; Colonic Neoplasms; Eczema; Infections; Kidney Calculi; Pain; Plague; Premature Birth; Rectal Neoplasms; Sepsis; Bacterial Infections; Eye Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Sleep Initiation and Maintenance Disorders; Anxiety; Dementia; Depressive Disorder; Schizophrenia
Unknown
Small molecule
Approved
OTHER
ORAL
Prostatic Neoplasms, Castration-Resistant; Carcinoma; Adrenal Cortex Neoplasms; Neoplasms
Cytochrome P450 11A1 inhibitor
Small molecule
Approved
OTHER
ORAL
Central Nervous System Neoplasms; Head and Neck Neoplasms; Arthritis, Rheumatoid; Cystinuria; Hepatolenticular Degeneration; Inflammation; Rheumatic Diseases; Spondylitis
Copper chelating agent
Small molecule
Approved
Unknown
Unknown
Sepsis; Vaginitis; Carcinoma, Non-Small-Cell Lung; Periapical Periodontitis; Prediabetic State; Severe Acute Respiratory Syndrome; Breast Neoplasms; Candidiasis, Vulvovaginal; Chorioretinitis; Hernia; Hernia, Ventral; Kidney Calculi; Malaria; Nasal Obstruction; Pain; Pneumonia, Pneumocystis; Skin Diseases; Staphylococcal Infections; Vaginosis, Bacterial; Acne Vulgaris; Bacterial Infections; Endometritis; Infections; Intraabdominal Infections; Osteomyelitis
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Unknown
Dopamine D2 receptor antagonist
Small molecule
Approved
OTHER
INJECTION
Sarcoma; Sarcoma, Ewing; Neoplasms
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Appendicitis; Cognitive Dysfunction; Fatigue; Head and Neck Neoplasms; Heart Arrest; Hemorrhoids; Marijuana Abuse; Mental Disorders; Multiple Sclerosis; Neural Tube Defects; Opioid-Related Disorders; Perceptual Disorders; Phobia, Social; Radius Fractures; Respiratory Insufficiency; Schizophrenia; Sepsis; Stroke; Substance-Related Disorders; Tobacco Use Disorder; Borderline Personality Disorder; Brain Injuries; Breast Neoplasms; Cancer Pain; Cataract; Child Development Disorders, Pervasive; Cocaine-Related Disorders; Complex Regional Pain Syndromes; Coronavirus Infections; Dental Anxiety; Depressive Disorder, Treatment-Resistant; Fractures, Multiple; Heart Septal Defects, Ventricular; Hypertrophy; Ischemic Stroke; Lung Neoplasms; Obsessive-Compulsive Disorder; Paget Disease, Extramammary; Parkinson Disease; Respiratory Distress Syndrome; Rett Syndrome; Severe Acute Respiratory Syndrome; Strabismus; Stress Disorders, Post-Traumatic; Subarachnoid Hemorrhage; Temporomandibular Joint Disorders; Alcoholism; Anemia, Sickle Cell; Bipolar Disorder; Chronic Pain; Delirium; Depression, Postpartum; Depressive Disorder; Depressive Disorder, Major; Epilepsy; Fractures, Bone; Headache; Lung Diseases; Mucositis; Neoplasms; Neuralgia; Obesity, Morbid; Pain; Pharyngitis; Postoperative Complications; Renal Colic; Rib Fractures; Shock, Septic; Spinal Stenosis; Status Asthmaticus; Status Epilepticus; Suicidal Ideation; Wounds and Injuries
Unknown
Small molecule
Approved
Unknown
Unknown
Polyuria; Urinary Incontinence
Unknown
Small molecule
Approved
Unknown
Unknown
Pain; Postoperative Nausea and Vomiting; Psychotic Disorders
D2-like dopamine receptor antagonist
Small molecule
Approved
Unknown
Unknown
Psychotic Disorders
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
INHALATION; ORAL
Amyotrophic Lateral Sclerosis; Asthma; Brain Injuries; Diabetic Retinopathy; Hypotension, Orthostatic; Tobacco Use Disorder; Tourette Syndrome; Albinism; Albinism, Oculocutaneous; Angelman Syndrome; Aphasia; Back Pain; Child Development Disorders, Pervasive; Chronic Pain; Cocaine-Related Disorders; Macular Degeneration; Pain; Retinitis Pigmentosa; Schizophrenia; Spinal Cord Injuries; Stress Disorders, Post-Traumatic; Amblyopia; Restless Legs Syndrome; Stroke; Parkinson Disease
Dopamine D3 receptor agonist
Small molecule
Approved
Unknown
Unknown
Analgesia; Hepatitis C; Intestinal Obstruction; Paget Disease, Extramammary; Diabetes Mellitus, Type 1; Diabetic Neuropathies; Feeding and Eating Disorders; Hypogonadism; Irritable Bowel Syndrome; Neuralgia; Obesity; Pruritus; Chronic Pain; Epilepsy; Heroin Dependence; Low Back Pain; Morphine Dependence; Mycosis Fungoides; Opioid-Related Disorders; Osteoarthritis; Pain; Parkinson Disease; Restless Legs Syndrome; Sezary Syndrome; Substance-Related Disorders; Substance Withdrawal Syndrome; Constipation
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
TOPICAL
Psoriasis; Breast Neoplasms; Dermatitis, Atopic; Hemorrhoids; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Hyperemia; Neoplasms; Common Cold; Conjunctivitis, Allergic; Influenza, Human; Respiratory Tract Diseases; Eye Manifestations; Nasal Obstruction
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Adrenal Cortex Neoplasms; Carcinoma in Situ; Dementia; Head and Neck Neoplasms; HIV Wasting Syndrome; Pulmonary Disease, Chronic Obstructive; Uterine Neoplasms; Breast Neoplasms; Endometrial Neoplasms; Hot Flashes; Liver Neoplasms; Acquired Immunodeficiency Syndrome; Anorexia; Cachexia; Neoplasms; Primary Immunodeficiency Diseases
Progesterone receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Astrocytoma; Brain Neoplasms; Carcinoma, Hepatocellular; Colorectal Neoplasms; Digestive System Neoplasms; Glioblastoma; Gliosarcoma; Neoplasms; Oligodendroglioma; Intracranial Hypertension; Meningitis, Cryptococcal; Candidiasis; Infections; Meningitis
Thymidylate synthase inhibitor
Small molecule
Approved
Unknown
Unknown
Infections; Bacteremia; Gram-Positive Bacterial Infections; Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
ORAL
HIV Infections; Osteomyelitis; Acquired Immunodeficiency Syndrome; Meningitis; Tuberculosis, Multidrug-Resistant; Tuberculosis; Tuberculosis, Pulmonary
70S ribosome inhibitor
Small molecule
Approved
DERMATOLOGY; OTHER
ORAL; TOPICAL
Amyotrophic Lateral Sclerosis; Autistic Disorder; Glioblastoma; Hematologic Neoplasms; Hypercholesterolemia; Myelodysplastic-Myeloproliferative Diseases; Neoplasms, Plasma Cell; Anemia; Anti-Neutrophil Cytoplasmic Antibody-Associated Vasculitis; Carcinoma, Adenoid Cystic; Cholangitis, Sclerosing; Colorectal Neoplasms; Emphysema; Keratosis, Actinic; Kidney Neoplasms; Lung Neoplasms; Lymphoma; Melanoma; Multiple Myeloma; Neuroblastoma; Pancreatic Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Severe Acute Respiratory Syndrome; Small Cell Lung Carcinoma; Striae Distensae; Breast Neoplasms; Carcinoma, Basal Cell; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Leukemia; Leukemia, Myeloid, Acute; Myelodysplastic Syndromes; Myeloproliferative Disorders; Purpura, Thrombocytopenic, Idiopathic; Rosacea; Skin Neoplasms; Acne Vulgaris; Hyperpigmentation; Leukemia, Promyelocytic, Acute; Melanosis; Neoplasms
Retinoic acid receptor agonist
Small molecule
Approved
Unknown
Unknown
Leukemia, Myeloid, Acute; Urinary Bladder, Overactive; Breast Neoplasms; Cellulitis; Dermatitis; Eczema; Staphylococcal Infections; Tuberculosis; Urinary Tract Infections; Cystic Fibrosis; Nasal Obstruction; Skin Diseases; Urinary Bladder Neoplasms; Bacterial Infections; Infections; Otitis Media; Prostatitis; Respiratory Tract Infections; Sprains and Strains
Bacterial penicillin-binding protein inhibitor