Display Options:
Total: 6532
Small molecule
Approved
OTHER
ORAL
Alcoholism; Brain Injuries; Chondrocalcinosis; Diabetes Mellitus; Diabetes Mellitus, Type 2; Influenza in Birds; Kidney Diseases; Neoplasms; Cellulitis; Heart Failure; Heart Failure, Systolic; Cystitis, Hemorrhagic; Infections; Infertility, Male; Obesity; Urinary Tract Infections; Gout
Solute carrier family 22 member 11 inhibitor
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Urinary Bladder, Neurogenic; Digestive System Diseases
Unknown
Small molecule
Approved
OTHER
TOPICAL
Dandruff; Dermatitis, Seborrheic; Pruritus; Tinea
Unknown
Small molecule
Approved
OTHER
ORAL
Epilepsy
Sodium channel alpha subunit blocker
Small molecule
Approved
OTHER
ORAL
Amphetamine-Related Disorders; Fatigue; HIV Infections; Multiple Myeloma; Neoplasms; Obesity; Prostatic Neoplasms, Castration-Resistant; Retinal Dystrophies; Sarcoma; Alcohol-Related Disorders; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Cocaine-Related Disorders; Glioblastoma; Melanoma; Neoplasms, Germ Cell and Embryonal; Opioid-Related Disorders; Pancreatic Neoplasms; Paraganglioma; Severe Acute Respiratory Syndrome; Alcoholism; Ectoparasitic Infestations
Aldehyde dehydrogenase inhibitor
Small molecule
Approved
Unknown
Unknown
Crohn Disease; Gastroparesis; Motion Sickness; Anxiety; Dementia; Depressive Disorder; Hyperemesis Gravidarum; Migraine with Aura; Migraine without Aura; Nausea; Pain; Schizophrenia; Vertigo; Vomiting; Hypersensitivity; Pruritus
Unknown
Small molecule
Approved
Unknown
Unknown
Hypoglycemia; Obesity; Sleep Apnea, Obstructive; Mydriasis; Presbyopia; Cardiovascular Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Hypertension; Hypotension, Orthostatic; Infections; Mucositis; Neoplasms; Obesity; Ocular Hypertension; Orthostatic Intolerance; Ovarian Cysts; Pain; Stomatitis; Vascular Diseases; Acute Lung Injury; Bronchiolitis; Cognitive Dysfunction; Mydriasis; Shock, Septic; Stress Disorders, Post-Traumatic; Common Cold; Eye Diseases; Fecal Incontinence; Hypotension; Influenza, Human; Ischemic Stroke; Respiratory Tract Infections; Rhinitis, Allergic, Seasonal; Stroke; Cardiovascular Diseases; Eye Manifestations; Hemorrhoids; Nasal Obstruction
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Melanoma; Osteomyelitis; Acquired Immunodeficiency Syndrome; Diabetic Foot; Tuberculosis, Multidrug-Resistant; Ulcer; Meningitis; HIV Infections; Silicosis; Tuberculosis; Tuberculosis, Pulmonary
Enoyl-[acyl-carrier-protein] reductase inhibitor
Small molecule
Approved
OTHER
FOR RX COMPOUNDING; INJECTION; ORAL; RECTAL; TOPICAL; VAGINAL
Diabetes Mellitus, Type 1; Fibromyalgia; HIV Infections; Infections; Insulin Resistance; Lymphoma, Large-Cell, Anaplastic; Obesity; Tobacco Use Disorder; Addison Disease; Adrenal Cortex Neoplasms; Aging; Atrial Fibrillation; Borderline Personality Disorder; Central Nervous System Neoplasms; Granuloma, Pyogenic; Heart Failure; Inflammatory Bowel Diseases; Leukemia, Mast-Cell; Lymphohistiocytosis, Hemophagocytic; Lymphoma, Large B-Cell, Diffuse; Melanoma; Memory Disorders; Multiple Myeloma; Myocardial Infarction; Neoplasms, Plasma Cell; Opioid-Related Disorders; Pancreatitis; Phobic Disorders; Wounds and Injuries; Alcoholism; Alopecia Areata; Anemia, Refractory; Anemia, Refractory, with Excess of Blasts; Bronchopulmonary Dysplasia; Eczema; Heart Arrest; Hypotension; Hypoxia; Influenza, Human; Leukemia, Biphenotypic, Acute; Leukemia, Erythroblastic, Acute; Leukemia, Lymphoid; Leukemia, Megakaryoblastic, Acute; Leukemia, Monocytic, Acute; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Acute; Leukemia, Myelomonocytic, Chronic; Liver Cirrhosis; Myelodysplastic Syndromes; Myeloproliferative Disorders; Oral Submucous Fibrosis; Pain; Pneumonia, Viral; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sepsis; Severe Acute Respiratory Syndrome; Shock, Septic; Adrenal Hyperplasia, Congenital; Adrenal Insufficiency; Arthritis, Juvenile; Arthritis, Psoriatic; Arthritis, Rheumatoid; Asthma; Bursitis; Colitis, Ulcerative; Conjunctivitis, Allergic; Crohn Disease; Dermatitis; Dermatitis, Atopic; Dermatitis, Seborrheic; Endocrine System Diseases; Exanthema; Eye Diseases; Hemorrhoids; Herpes Labialis; Inflammation; Leukemia; Lymphoma; Nasal Obstruction; Neoplasms; Osteoarthritis; Otitis Externa; Pneumonia; Pruritus; Psoriasis; Serum Sickness; Skin Diseases; Spondylitis; Tenosynovitis
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
TOPICAL
Unknown
Tyrosinase inhibitor
Small molecule
Approved
Unknown
Unknown
Glucosephosphate Dehydrogenase Deficiency; Obesity; Severe Acute Respiratory Syndrome; Malaria, Falciparum; Malaria, Vivax; Pneumonia, Pneumocystis; Malaria
Unknown
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases; Mydriasis; Prostatic Neoplasms, Castration-Resistant; Pheochromocytoma
Adrenergic receptor alpha antagonist
Small molecule
Approved
Unknown
Unknown
Arthritis, Rheumatoid; Glioblastoma; Neoplasm Metastasis; Adenocarcinoma; Asperger Syndrome; Autistic Disorder; Biliary Tract Diseases; Biliary Tract Neoplasms; Carcinoma, Neuroendocrine; Child Development Disorders, Pervasive; Colonic Neoplasms; Esophageal Neoplasms; Neoplasms; Osteosarcoma; Uterine Neoplasms; Carcinoma, Hepatocellular; Carcinoma, Pancreatic Ductal; Colorectal Neoplasms; Depressive Disorder; Down Syndrome; Liver Neoplasms; Nasopharyngeal Carcinoma; Pancreatic Neoplasms; Psychotic Disorders; Rectal Neoplasms; Schizophrenia; Stomach Neoplasms
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Osteomyelitis; Psoriasis; Rheumatic Heart Disease; HIV Infections; Syphilis; Bacterial Infections; Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Bradycardia; Myalgia; Stroke
Unknown
Small molecule
Approved
Unknown
Unknown
Anemia, Sickle Cell; Constipation; Neck Pain; Osteoarthritis; Myopia; Toothache; Cough; Pain
Unknown
Small molecule
Approved
Unknown
Unknown
Pain
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Bacterial Infections; Cystitis; Urinary Tract Infections
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Amyotrophic Lateral Sclerosis; Gangliosidoses, GM2; Head and Neck Neoplasms; Leukemia, Lymphocytic, Chronic, B-Cell; Myelodysplastic Syndromes; Sandhoff Disease; Tay-Sachs Disease; Toxoplasmosis, Cerebral; Anemia; Chorioretinitis; Depressive Disorder; HIV Infections; Malaria, Falciparum; Malaria, Vivax; Pneumonia, Pneumocystis; Pregnancy; Premature Birth; Schistosomiasis; Schizophrenia; Toxoplasmosis, Congenital; Malaria; Toxoplasmosis
Dihydrofolate reductase inhibitor
Small molecule
Approved
OTHER
INJECTION
Unknown
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Anemia; Cocaine-Related Disorders; Immune System Diseases; Leukemia; Lymphoma; Neuroblastoma; Anemia, Sickle Cell; Optic Neuritis; Pancreatic Neoplasms; Polyneuropathies; Thalassemia; Wounds and Injuries; Anxiety; Dementia; Depressive Disorder; Schizophrenia; Epilepsy; Seizures
Sodium channel alpha subunit blocker
Small molecule
Approved
OTHER
ORAL
Osteomyelitis; Bacterial Infections; Eye Infections
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
Unknown
Unknown
Hernias, Diaphragmatic, Congenital; Paraganglioma; Pheochromocytoma; Cardiovascular Diseases
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Urinary Bladder, Overactive; Peptic Ulcer
Muscarinic acetylcholine receptor M1 antagonist
Small molecule
Approved
OTHER
INJECTION; SUBCUTANEOUS
Muscular Dystrophy, Facioscapulohumeral; HIV Wasting Syndrome; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Pulmonary Disease, Chronic Obstructive; Weight Loss; Hypogonadism; Neoplasms; Orchitis
Androgen Receptor agonist
Small molecule
Approved
OTHER
ORAL; SUBLINGUAL
Dementia, Vascular; Fragile X Syndrome; Cardiovascular Diseases
Adrenergic receptor alpha antagonist
Small molecule
Approved
Unknown
Unknown
Lung Neoplasms; Polycystic Kidney Diseases; Rectal Neoplasms; Breast Neoplasms; Cardiovascular Diseases; Cerebral Hemorrhage; Heart Diseases; Heart Failure; Neoplasms; Pre-Eclampsia; Stroke; Vascular Diseases; Atherosclerosis; Coronary Disease; Diabetes Mellitus, Type 2; Hypercholesterolemia; Ovarian Neoplasms; Uterine Cervical Neoplasms; Hypertension
Unknown
Small molecule
Approved
OTHER
ORAL
Burkitt Lymphoma; Astrocytoma; Blastic Plasmacytoid Dendritic Cell Neoplasm; Brain Neoplasms; Colitis; Glioblastoma; Glioma; Oligodendroglioma; Colitis, Ulcerative; Crohn Disease; Histiocytosis, Langerhans-Cell; Leukemia; Leukemia, Biphenotypic, Acute; Leukemia, Myeloid, Acute; Leukemia, Promyelocytic, Acute; Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Leukemia, Lymphoid; Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma
Amidophosphoribosyltransferase inhibitor
Small molecule
Approved
OTHER
ORAL
Unknown
Bacterial dihydropteroate synthase inhibitor
Small molecule
Approved
OTHER
ORAL
Andersen Syndrome; Diabetes Mellitus, Type 1; Hypotension, Orthostatic; Melanoma; Prostatic Neoplasms, Castration-Resistant; Psychotic Disorders; Schizophrenia; Small Cell Lung Carcinoma; Chronic Pain; Cysticercosis; Helicobacter Infections; Hypertension, Pulmonary; Kidney Diseases; Landau-Kleffner Syndrome; Macular Edema; Multiple Sclerosis; Retinoschisis; Sleep Apnea, Obstructive; Status Epilepticus; Stroke; Apnea; Carcinoma, Hepatocellular; Hydrocephalus, Normal Pressure; Pseudotumor Cerebri; Altitude Sickness; Edema; Epilepsy; Glaucoma; Glaucoma, Angle-Closure; Heart Failure; Seizures
Carbonic anhydrase II inhibitor
Small molecule
Approved
OTHER
ORAL
Unknown
Muscarinic acetylcholine receptor M1 antagonist