Display Options:
Total: 6532
Small molecule
Approved
OTHER
ORAL
Depressive Disorder, Major; Substance Withdrawal Syndrome; Alcoholism; Anxiety; Anxiety Disorders
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Glaucoma
Acetylcholinesterase inhibitor
Small molecule
Approved
OTHER
OPHTHALMIC
Unknown
Acetylcholinesterase inhibitor
Small molecule
Approved
OTHER
OPHTHALMIC
Ocular Hypertension; Parkinson Disease; Presbyopia; Sialorrhea; Eye Diseases; Mydriasis
Muscarinic acetylcholine receptor M3 antagonist
Small molecule
Approved
Unknown
Unknown
Glaucoma; Hypertension
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
INTRAMUSCULAR
Hypoglycemia; Hypotension, Orthostatic; Insulin Resistance; Orthostatic Intolerance; Postoperative Complications; Prediabetic State; Amyotrophic Lateral Sclerosis; Blood Coagulation Disorders; Bradycardia; Breast Neoplasms; Heart Arrest; Hemorrhage; Hypospadias; Organophosphate Poisoning; Pneumonia, Ventilator-Associated; Rhinitis, Allergic, Seasonal; Amblyopia; Anisometropia; Dwarfism, Pituitary; Headache; Myopia; Myopia, Degenerative; Pain; Strabismus; Digestive System Diseases; Mydriasis; Poisoning
Muscarinic acetylcholine receptor M1 antagonist
Small molecule
Approved
OTHER; PEDIATRICS; RESPIRATORY
DENTAL; INHALATION; INJECTION; INTRA-ARTICULAR; INTRAMUSCULAR; INTRAVITREAL; NASAL; SUSPENSION; TOPICAL
Fibroma; Hearing Loss; Mucositis; Neuroma, Acoustic; Papilledema; Rotator Cuff Injuries; Tendon Entrapment; Alopecia Areata; Breast Neoplasms; Cataract; Complex Regional Pain Syndromes; Dermatitis, Atopic; Glaucoma; Hand Dermatoses; Humeral Fractures; Keloid; Lichen Planus; Pemphigoid, Benign Mucous Membrane; Psoriasis; Shoulder Pain; Ulnar Neuropathies; Uveal Melanoma; Uveomeningoencephalitic Syndrome; Vitiligo; Wet Macular Degeneration; Chalazion; Choroidal Neovascularization; Cough; Cystitis, Interstitial; Diabetic Retinopathy; Dupuytren Contracture; Eye Injuries; Lichen Planus, Oral; Macular Degeneration; Macular Edema; Optic Neuropathy, Ischemic; Osteoarthritis, Hip; Osteoarthritis, Knee; Otitis Media with Effusion; Pemphigus; Radiculopathy; Retinal Vein Occlusion; Rhinitis; Tendinopathy; Uveitis; Vitreoretinopathy, Proliferative; Anemia; Arthritis, Gouty; Arthritis, Rheumatoid; Asthma; Bursitis; Dermatitis; Multiple Sclerosis; Mycoses; Nasal Obstruction; Osteoarthritis; Pain; Rhinitis, Allergic, Seasonal; Serum Sickness; Skin Diseases; Tennis Elbow; Tenosynovitis; Tuberculosis, Pulmonary; Wounds and Injuries
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
INJECTION; ORAL
Amphetamine-Related Disorders; Hypertension, Pulmonary; Cocaine-Related Disorders; Substance-Related Disorders; Vascular Diseases; Atherosclerosis; Cardiovascular Diseases; Cerebrovascular Disorders; Coronary Disease; Diabetes Mellitus, Type 2; Heart Diseases; Hypercholesterolemia; Hypertension
Synaptic vesicular amine transporter inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Mu opioid receptor agonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Alcoholism; Chorioretinitis; Diabetes Mellitus; Diabetic Nephropathies; Dry Eye Syndromes; Leukemia; Leukemia, Myeloid, Acute; Melanosis; Non-alcoholic Fatty Liver Disease; Arrhythmogenic Right Ventricular Dysplasia; Cardiomyopathies; Cerebral Hemorrhage; Fatty Liver; Hypertension, Pulmonary; Macular Degeneration; Neoplasms; Neuroblastoma; Polycystic Ovary Syndrome; Puberty, Precocious; Severe Acute Respiratory Syndrome; Acne Vulgaris; Acute Kidney Injury; Aortic Valve Stenosis; Arthritis, Rheumatoid; Atrial Fibrillation; Heart Failure, Diastolic; Muscular Dystrophy, Duchenne; Non-ST Elevated Myocardial Infarction; Polycystic Kidney, Autosomal Dominant; Renal Insufficiency, Chronic; ST Elevation Myocardial Infarction; Ascites; Cardiovascular Diseases; Edema; Essential Hypertension; Fibrosis; Heart Failure; Hyperaldosteronism; Hypertension; Liver Cirrhosis; Myocardial Infarction; Nephrotic Syndrome; Toxemia
Mineralocorticoid receptor antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Pain
Sodium channel alpha subunit blocker
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
Dopamine D2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Psychotic Disorders
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
GABA-A receptor; anion channel positive modulator
Small molecule
Approved
MUSCULOSKELETAL; OTHER; RHEUMATOLOGY
ORAL
Liver Cirrhosis; Neoplasms; Peripheral Arterial Disease; Urogenital Neoplasms; Acute Coronary Syndrome; Amyotrophic Lateral Sclerosis; Atherosclerosis; Behcet Syndrome; Cholangiocarcinoma; Coronavirus Infections; Diabetic Nephropathies; Heart Diseases; Hepatitis C, Chronic; Hypertension; Intracranial Hemorrhages; Osteoarthritis, Knee; Pneumonia, Viral; Prostatic Neoplasms, Castration-Resistant; Renal Insufficiency, Chronic; Stomatitis, Aphthous; Vascular Diseases; Arrhythmias, Cardiac; Asthma; Atrial Fibrillation; Cardiovascular Diseases; Coronary Disease; Heart Failure; Liver Cirrhosis, Biliary; Lung Diseases; Multiple Myeloma; Myocardial Infarction; Non-ST Elevated Myocardial Infarction; Pericarditis; Postpericardiotomy Syndrome; Reperfusion Injury; Severe Acute Respiratory Syndrome; ST Elevation Myocardial Infarction; Vasculitis; Vitreoretinopathy, Proliferative; Familial Mediterranean Fever; Gout
Tubulin inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Estrogen receptor alpha agonist
Small molecule
Approved
Unknown
Unknown
Biliary Dyskinesia; Bursitis; Diabetes Mellitus; Digestive System Diseases; Inflammatory Bowel Diseases; Intervertebral Disc Displacement; Lung Diseases, Interstitial; Paget Disease, Extramammary; Peripheral Nervous System Diseases; Rosacea; Anxiety; Cystitis, Interstitial; Dementia; Depressive Disorder, Major; Fibromyalgia; Headache; Migraine Disorders; Neuralgia; Pain; Schizophrenia; Sleep Initiation and Maintenance Disorders; Depressive Disorder
Unknown
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Hernia, Inguinal; Hypersensitivity
Unknown
Small molecule
Approved
OTHER; PEDIATRICS
INHALATION; INJECTION; INTRAMUSCULAR; INTRAVENOUS; ORAL
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Depressive Disorder; Depressive Disorder, Major
Monoamine oxidase inhibitor
Small molecule
Approved
Unknown
Unknown
Severe Acute Respiratory Syndrome; Asthma; Hyperhidrosis; Pulmonary Disease, Chronic Obstructive
Unknown
Small molecule
Approved
OTHER
INJECTION
Unknown
Dopamine D2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Stroke; Abdominal Pain; Alcoholism; Mitral Valve Insufficiency; Severe Acute Respiratory Syndrome; Hypersensitivity
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Progesterone receptor agonist
Small molecule
Approved
OTHER
ORAL; TOPICAL
Adenoma; Hypospadias; Oral Ulcer; Bronchiolitis; Dermatitis, Atopic; Dry Eye Syndromes; Glaucoma; Hyaline Membrane Disease; Macular Edema; Melanoma; Neck Pain; Respiratory Distress Syndrome, Newborn; Retinal Vein Occlusion; Sciatica; Tachypnea; Carpal Tunnel Syndrome; Cough; Eczema; Gout; Hypersensitivity; Lichen Planus, Oral; Orbital Pseudotumor; Pharyngitis; Pregnancy; Premature Birth; Psoriasis; Respiratory Distress Syndrome; Rhinitis, Allergic, Seasonal; Eye Diseases; Hemorrhoids; Lung Diseases, Obstructive; Nasal Obstruction
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Cough
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
HIV Infections; Hypertension; IgA Vasculitis; Anemia, Sickle Cell; Arthritis, Rheumatoid; Carotid Stenosis; Ovarian Neoplasms; Pancreatic Neoplasms; Angina, Stable; Cardiovascular Diseases; Heart Diseases; Myocardial Ischemia; Severe Acute Respiratory Syndrome; Coronary Artery Disease; Stroke; Thrombosis
3',5'-cyclic phosphodiesterase inhibitor
Small molecule
Approved
OTHER
ORAL
Chronic Pain; Endotoxemia; Hepatitis C, Chronic; Lymphoma; Neoplasms; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker