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Total: 6532
Small molecule
Approved
CARDIOVASCULAR; DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Diabetes Mellitus, Type 2; Glioblastoma; Hypertension, Pulmonary; Neoplasms; Primary Myelofibrosis; Heart Diseases; Pneumonia; Severe Acute Respiratory Syndrome; Cardiovascular Diseases; Collagen Diseases; Diabetic Nephropathies; Diabetic Retinopathy; Heart Failure; Hypertension; Myocardial Infarction; Renal Insufficiency; Ventricular Dysfunction, Left
Angiotensin-converting enzyme inhibitor
Small molecule
Approved
Unknown
Unknown
Anemia; HIV Infections; Malaria; Malaria, Falciparum; Malaria, Vivax; Pneumonia, Pneumocystis; Pregnancy; Premature Birth
Dihydropteroate synthetase inhibitor
Small molecule
Approved
Unknown
Unknown
Attention Deficit Disorder with Hyperactivity; Cystic Fibrosis; Coronary Disease; Demyelinating Diseases; Hyperparathyroidism, Primary; Migraine with Aura; Multiple Sclerosis, Chronic Progressive; Optic Neuritis; Hypertension; Cardiovascular Diseases
Unknown
Small molecule
Approved
CARDIOVASCULAR; OTHER; UROLOGY AND KIDNEY
INJECTION; URETHRAL
Arteriosclerosis Obliterans; Optic Neuropathy, Ischemic; Peripheral Arterial Disease; Peripheral Vascular Diseases; Respiratory Distress Syndrome; Severe Acute Respiratory Syndrome; Sexual Dysfunction, Physiological; Heart Failure; Macular Degeneration; Prostatic Neoplasms, Castration-Resistant; Cardiovascular Diseases; Ductus Arteriosus, Patent; Erectile Dysfunction
Prostanoid EP1 receptor agonist
Small molecule
Approved
OTHER
INJECTION; TOPICAL
Leukemia; Myopia; Neoplasm Metastasis; Renal Insufficiency, Chronic; Urethral Stricture; Appendiceal Neoplasms; Biliary Tract Neoplasms; Carcinoma, Squamous Cell; Cholangiocarcinoma; Cholangitis, Sclerosing; Corneal Opacity; Esophageal Stenosis; Glaucoma, Neovascular; Glaucoma, Open-Angle; Keratoconus; Liver Neoplasms; Pterygium; Sarcoma; Anus Neoplasms; Breast Neoplasms; Carcinoma; Carcinoma, Hepatocellular; Carcinoma in Situ; Carcinoma, Non-Small-Cell Lung; Carcinoma, Transitional Cell; Colorectal Neoplasms; Head and Neck Neoplasms; Lung Neoplasms; Mesothelioma; Nasopharyngeal Neoplasms; Pancreatic Neoplasms; Stomach Neoplasms; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Adenocarcinoma; Glaucoma; Neoplasms
DNA inhibitor
Small molecule
Unknown
Unknown
Unknown
Cardiovascular Diseases; Hodgkin Disease; Atrial Fibrillation; Heart Failure; Arrhythmias, Cardiac; Diabetes Mellitus; Hypertension
Voltage-gated L-type calcium channel blocker
Small molecule
Approved
OTHER
ORAL
Anxiety
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
OTHER
ORAL
Multiple Sclerosis; Sunburn; Angioedema; Conjunctivitis, Allergic; Hypersensitivity; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; Rhinitis, Vasomotor; Urticaria
Histamine H1 receptor antagonist
Small molecule
Approved
IMMUNE SYSTEM; OTHER
ORAL; TOPICAL
Glioblastoma; Insulin Resistance; Alzheimer Disease; Asthma; Diabetes Mellitus, Type 2; Erectile Dysfunction; Essential Hypertension; Gastroparesis; Hepatitis C; Immune System Diseases; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma; Lymphoma, Non-Hodgkin; Melanoma; Multiple Sclerosis; Nausea; Neuroblastoma; Osteoporosis; Premature Birth; Pulmonary Disease, Chronic Obstructive; Breast Neoplasms; Burns; Hypogonadism; Neoplasms; Prostatic Neoplasms; Psoriasis; Acne Vulgaris; Candidiasis, Vulvovaginal; Dermatitis; Prostatic Neoplasms, Castration-Resistant; Respiratory Distress Syndrome; Vaginosis, Bacterial; Adrenal Gland Diseases; Blastomycosis; Dermatitis, Seborrheic; Onychomycosis; Tinea; Tinea Pedis
Cytochrome P450 51 inhibitor
Small molecule
Approved
Unknown
Unknown
Osteomyelitis
Bacterial penicillin-binding protein inhibitor
Small molecule
Unknown
Unknown
Unknown
Amyotrophic Lateral Sclerosis; Depression; Depressive Disorder; Depressive Disorder, Major
Serotonin 2a (5-HT2a) receptor antagonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Appendicitis; Peritonitis; Sepsis; Bacterial Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Adrenal Hyperplasia, Congenital; Substance-Related Disorders; Anus Diseases; Epilepsies, Partial; Fissure in Ano; Proteinuria; Renal Insufficiency, Chronic; Diabetic Nephropathies; Hypertension, Pulmonary; Kidney Calculi; Myocardial Ischemia; Placenta Previa; Premature Birth; Raynaud Disease; Cardiovascular Diseases; Coronary Vasospasm; Hypertension
Voltage-gated L-type calcium channel blocker
Small molecule
Unknown
Unknown
Unknown
Hepatitis C; Anemia, Sickle Cell; Carcinoma, Squamous Cell; Depressive Disorder; Rotator Cuff Injuries; Stress Disorders, Post-Traumatic; Toothache; Back Pain; Cocaine-Related Disorders; Depressive Disorder, Major; Heroin Dependence; HIV Infections; Intervertebral Disc Degeneration; Low Back Pain; Morphine Dependence; Neonatal Abstinence Syndrome; Neuralgia; Osteoarthritis; Substance Withdrawal Syndrome; Acute Pain; Chronic Pain; Drug Overdose; Opioid-Related Disorders; Pain; Substance-Related Disorders
Kappa opioid receptor agonist
Small molecule
Approved
Unknown
Unknown
Sleep Apnea, Obstructive; Alcoholism; Diabetic Neuropathies; Alzheimer Disease; Anxiety; Dementia; Depressive Disorder, Major; Schizophrenia; Sleep Initiation and Maintenance Disorders; Sleep Wake Disorders; Depressive Disorder
Unknown
Small molecule
Approved
OTHER
INJECTION
Breast Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Hypotension, Orthostatic; Orthostatic Intolerance; Depressive Disorder; Hypotension; Myocardial Infarction; Hypertension
Unknown
Small molecule
Approved
CARDIOVASCULAR; GASTROINTESTINAL; OTHER
INJECTION; INTRA-ANAL; SUBLINGUAL; TRANSDERMAL
Colorectal Neoplasms; Hypotension; Peripheral Arterial Disease; Hypertension, Pulmonary; Infections; Inflammation; Phlebitis; Rectal Neoplasms; Carcinoma, Non-Small-Cell Lung; Diabetic Neuropathies; Erectile Dysfunction; Hot Flashes; Lung Neoplasms; Shock; Tendinopathy; Arthritis, Rheumatoid; Bone Diseases, Metabolic; Muscle Cramp; Myocardial Ischemia; Osteoporosis; Raynaud Disease; Reperfusion Injury; Scleroderma, Localized; Stroke; Wounds and Injuries; Angina Pectoris; Angina, Stable; Cardiovascular Diseases; Coronary Artery Disease; Coronary Disease; Heart Failure; Hemorrhoids; Hypertension; Myocardial Infarction; Pain
Soluble guanylate cyclase activator
Small molecule
Approved
Unknown
Unknown
Hypersensitivity
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Osteoporosis; Stress Disorders, Post-Traumatic; Atrial Fibrillation; Cerebrovascular Disorders; Essential Hypertension; Heart Diseases; Heart Failure; Hemangioma; Hypertrophy, Left Ventricular; Marfan Syndrome; Mitral Valve Stenosis; Myocardial Ischemia; Angina Pectoris; Angina, Stable; Cardiovascular Diseases; Coronary Artery Disease; Diabetes Mellitus; Hypertension; Myocardial Infarction; Stroke
Beta-1 adrenergic receptor antagonist
Small molecule
Approved
OTHER
INHALATION; NASAL
Rhinitis, Allergic, Perennial; Asthma; Lung Diseases, Obstructive; Nasal Obstruction; Rhinitis
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
ORAL
Unknown
Adrenergic receptor alpha antagonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Hypertension
Unknown
Small molecule
Unknown
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Renal Colic; Osteoarthritis, Knee; Tennis Elbow; Arthralgia; Arthritis, Rheumatoid; Eye Diseases; Myalgia; Osteoarthritis; Rheumatic Diseases
Cyclooxygenase inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Bipolar Disorder; Cystic Fibrosis; Depressive Disorder, Major; Pulmonary Disease, Chronic Obstructive; Obesity; Brain Injuries; Brain Ischemia; Delirium; Hypothermia; Obsessive-Compulsive Disorder; Panic Disorder; Coronary Disease
Unknown
Small molecule
Approved
Unknown
Unknown
Multiple Sclerosis, Relapsing-Remitting
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Bacterial Infections
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
GABA-A receptor; anion channel positive allosteric modulator
Small molecule
Approved
OTHER; PREGNANCY AND GYNECOLOGY
IMPLANTATION; INTRAUTERINE; ORAL
Diabetes Mellitus, Type 2; Hepatitis B, Chronic; Hepatitis C, Chronic; Leukemia, Lymphocytic, Chronic, B-Cell; Neoplasms; Non-alcoholic Fatty Liver Disease; Adenomyosis; HIV Infections; Ovarian Neoplasms; Pain; Anorexia Nervosa; Bone Diseases, Metabolic; Dysmenorrhea; Endometrial Hyperplasia; Endometriosis; Hemorrhage; Migraine Disorders; Menorrhagia
Progesterone receptor agonist