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Total: 10647
Small molecule
Approved
OTHER
ORAL
Cardiovascular Diseases; Hypertension
Voltage-gated L-type calcium channel blocker
Small molecule
Approved
OTHER
ORAL
Glioblastoma; Vascular Diseases; Breast Neoplasms; Cocaine-Related Disorders; Epilepsy; Esophageal and Gastric Varices; Hypertension, Pulmonary; Hypoglycemia; Kidney Diseases; Lymphoma; Neoplasms; Prostatic Neoplasms, Castration-Resistant; Stress Disorders, Post-Traumatic; Tobacco Use Disorder; Atherosclerosis; Atrial Fibrillation; Coronary Disease; Diabetes Mellitus, Type 2; Essential Hypertension; Hypercholesterolemia; Hypertension, Portal; Hypertrophy, Left Ventricular; Leukemia, Lymphoid; Leukemia, Myeloid, Acute; Multiple Myeloma; Cardiovascular Diseases; Heart Failure; Hypertension; Myocardial Infarction; Ventricular Dysfunction, Left
Adrenergic receptor alpha-1 antagonist
Small molecule
Approved
DERMATOLOGY; OTHER
TOPICAL
Dermatitis, Perioral; Dermatitis, Seborrheic; Acne Vulgaris; Erythema; Rosacea
Unknown
Small molecule
Approved
CARDIOVASCULAR; OTHER
INJECTION
Unknown
HERG blocker
Small molecule
Unknown
Unknown
Unknown
Pre-Eclampsia; Pancreatic Neoplasms; Carcinoma, Pancreatic Ductal; Eosinophilic Esophagitis; Non-alcoholic Fatty Liver Disease; Essential Hypertension; Hypertrophy, Left Ventricular; Marfan Syndrome; Hypertension; Kidney Diseases; Kidney Failure, Chronic; Proteinuria; Stroke
Type-1 angiotensin II receptor antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Atherosclerosis; Coronary Disease; Hypercholesterolemia; Hypertension; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
DERMATOLOGY
ORAL
Osteomyelitis; Bacterial Infections
Bacterial 70S ribosome inhibitor
Small molecule
Approved
Unknown
Unknown
Anemia, Sickle Cell; Barrett Esophagus; Cardiovascular Diseases; Diabetic Retinopathy; Pulmonary Disease, Chronic Obstructive; Thoracic Neoplasms; Anxiety Disorders; Breast Carcinoma In Situ; Depressive Disorder, Major; Diabetes Insipidus; Head and Neck Neoplasms; HIV Infections; Li-Fraumeni Syndrome; Liver Diseases; Multiple Sclerosis; Muscular Dystrophy, Duchenne; Neuralgia; Osteoarthritis; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Sleep Apnea, Obstructive; Adenocarcinoma; Adenocarcinoma, Bronchiolo-Alveolar; Adenocarcinoma of Lung; Adenomatous Polyposis Coli; Aortic Aneurysm, Abdominal; Arthritis, Rheumatoid; Atrial Fibrillation; Bardet-Biedl Syndrome; Blindness; Breast Neoplasms; Burns; Carcinoma; Carcinoma, Hepatocellular; Carcinoma, Large Cell; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Cerebral Palsy; Colitis, Ulcerative; Colonic Neoplasms; Diabetic Foot; Endometrial Hyperplasia; Esophageal Neoplasms; Fragile X Syndrome; Frontotemporal Dementia; Geographic Atrophy; Glioblastoma; Heart Failure, Systolic; Hemangiosarcoma; Hepatitis; HIV-Associated Lipodystrophy Syndrome; Hypertension, Pulmonary; Intellectual Disability; Leukemia, Lymphocytic, Chronic, B-Cell; Low Back Pain; Lung Neoplasms; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Melanoma; Multiple Myeloma; Neoplasms; Neurobehavioral Manifestations; Neuroendocrine Tumors; Non-alcoholic Fatty Liver Disease; Ovarian Neoplasms; Pancreatic Neoplasms; Periodontitis; Peripheral Nervous System Diseases; Pregnancy; Prostatic Neoplasms; Rectal Neoplasms; Renal Insufficiency, Chronic; Severe Acute Respiratory Syndrome; Sex Chromosome Disorders of Sex Development; Small Cell Lung Carcinoma; Squamous Cell Carcinoma of Head and Neck; Triple Negative Breast Neoplasms; Urinary Bladder Neoplasms; Urogenital Neoplasms; Uterine Cervical Neoplasms; Weight Gain; Aging; Atherosclerosis; Bipolar Disorder; Brain Neoplasms; Cognitive Dysfunction; Colorectal Neoplasms; Coronary Disease; Diabetes, Gestational; Diabetes Mellitus, Type 1; Diabetes Mellitus, Type 2; Endometrial Neoplasms; Fatty Liver; Glucose Intolerance; Hidradenitis Suppurativa; Huntington Disease; Hypercholesterolemia; Hypertension; Infertility; Insulin Resistance; Lipid Metabolism Disorders; Liver Neoplasms; Metabolic Diseases; Metabolic Syndrome; Migraine Disorders; Muscular Dystrophies; Obesity; Peripheral Arterial Disease; Polycystic Kidney, Autosomal Dominant; Polycystic Ovary Syndrome; Prediabetic State; Prostatic Neoplasms, Castration-Resistant; Psoriasis; Psychotic Disorders; Schizophrenia; Diabetes Mellitus
Unknown
Small molecule
Approved
IMMUNE SYSTEM
ORAL
Hookworm Infections; Trichuriasis; Cysticercosis; Ectoparasitic Infestations; Elephantiasis, Filarial; Filariasis; HIV Infections; Malaria; Malnutrition; Onchocerciasis; Strongyloidiasis; Toxocariasis; Helminthiasis; Infections; Neurocysticercosis
Tubulin inhibitor
Small molecule
Approved
GASTROINTESTINAL; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
INJECTION; INTRAVENOUS
Osteomyelitis; Gram-Negative Bacterial Infections; Pancreatitis; Respiratory Insufficiency; Communicable Diseases; Tuberculosis; Tuberculosis, Pulmonary; Enterobacteriaceae Infections; Neonatal Sepsis; Pneumonia; Pneumonia, Bacterial; Pneumonia, Ventilator-Associated; Pyelonephritis; Sepsis; Shock, Septic; Bacteremia; Bacterial Infections; Infections; Intraabdominal Infections; Meningitis; Meningitis, Bacterial; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
Unknown
Unknown
Melanoma; Muscle Spasticity; Pain
Unknown
Small molecule
Approved
Unknown
Unknown
Tinea Pedis
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Cardiovascular Diseases; Heart Failure; Hypertension; Myocardial Infarction; Ventricular Dysfunction, Left
Angiotensin-converting enzyme inhibitor
Small molecule
Approved
OTHER
INTRAMUSCULAR; ORAL
Dyskinesia, Drug-Induced; Lecithin Cholesterol Acyltransferase Deficiency; Mood Disorders; Weight Loss; Amyotrophic Lateral Sclerosis; Anorexia Nervosa; Autistic Disorder; Delirium; Vomiting; Alcoholism; Anxiety; Borderline Personality Disorder; Dementia; Depressive Disorder; Depressive Disorder, Treatment-Resistant; Developmental Disabilities; Feeding and Eating Disorders; Gambling; Genital Neoplasms, Female; Huntington Disease; Intellectual Disability; Nausea; Neoplasms; Postoperative Nausea and Vomiting; Weight Gain; Bipolar Disorder; Depressive Disorder, Major; Psychomotor Agitation; Psychotic Disorders; Schizophrenia
D2-like dopamine receptor antagonist
Small molecule
Approved
OTHER
ORAL
Prostatic Neoplasms, Castration-Resistant; Neoplasms; Prostatic Neoplasms
Androgen Receptor antagonist
Small molecule
Approved
Unknown
Unknown
Stress Disorders, Post-Traumatic; Fasciitis, Plantar; Hernia, Inguinal; Rib Fractures; Appendicitis; Hallux Valgus; Joint Diseases; Leiomyoma; Osteoarthritis; Rotator Cuff Injuries; Shoulder Pain; Abdominal Pain; Breast Neoplasms; Chronic Pain; Hypotension; Knee Injuries; Neoplasms; Ovarian Cysts; Ovarian Neoplasms; Pain; Paralysis; Stomach Neoplasms
Unknown
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER; PEDIATRICS
ORAL
Feeding and Eating Disorders; Bulimia Nervosa; Cognitive Dysfunction; Hernias, Diaphragmatic, Congenital; Liver Diseases; Alcohol Drinking; Amphetamine-Related Disorders; Brain Ischemia; Diabetes Mellitus; Marijuana Abuse; Multiple Sclerosis; Parkinson Disease; Sciatica; Stress Disorders, Post-Traumatic; Alcoholism; Anxiety; Bipolar Disorder; Bulimia; Cocaine-Related Disorders; Dementia; Depressive Disorder; Diabetes Mellitus, Type 2; Epilepsies, Partial; Epilepsy, Tonic-Clonic; Essential Tremor; Gambling; Headache; Hyperlipidemias; Hypertension; Hypertriglyceridemia; Metabolic Syndrome; Obesity; Obsessive-Compulsive Disorder; Pain; Prader-Willi Syndrome; Schizophrenia; Smoking Cessation; Tobacco Use Disorder; Tourette Syndrome; Epilepsy; Lennox Gastaut Syndrome; Migraine Disorders; Seizures
Carbonic anhydrase II inhibitor
Small molecule
Approved
IMMUNE SYSTEM; OTHER
DENTAL; TOPICAL
Stomatitis; Lung Diseases, Obstructive
Phosphodiesterase 4 inhibitor
Small molecule
Approved
OTHER; RESPIRATORY
ORAL
Inflammation; Anemia, Sickle Cell; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Acne Vulgaris; Idiopathic Pulmonary Fibrosis; Lung Neoplasms; Tobacco Use Disorder; Pulmonary Disease, Chronic Obstructive; Asthma
Arachidonate 5-lipoxygenase inhibitor
Small molecule
Approved
OTHER
ORAL
HIV Infections; Alzheimer Disease; Dermatitis; Melanoma; Psoriasis
Retinoid receptor agonist
Small molecule
Approved
OTHER; RESPIRATORY
ORAL
Breast Neoplasms; Ovarian Neoplasms; Asthma; Lung Diseases, Obstructive
Cysteinyl leukotriene receptor 1 antagonist
Enzyme
Approved
Unknown
Unknown
Hepatitis C; HIV Infections
Polypeptides hydrolytic enzyme
Unknown
Approved
OTHER
INJECTION
Acute Kidney Injury
Diagnostic agent
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Breast Neoplasms; Obesity; Substance-Related Disorders; Cocaine-Related Disorders; Endometriosis; Infertility; Paget Disease, Extramammary; Pituitary ACTH Hypersecretion; Acromegaly; Diabetes Mellitus; Ovarian Hyperstimulation Syndrome; Restless Legs Syndrome; Parkinson Disease; Pituitary Neoplasms
Dopamine D2 receptor agonist
Small molecule
Approved
Unknown
Unknown
Status Epilepticus; Epilepsy
Unknown
Small molecule
Approved
RESPIRATORY
ORAL
Osteomyelitis; Bacterial Infections
Bacterial DNA gyrase inhibitor
Small molecule
Approved
EYE; OTHER; UROLOGY AND KIDNEY
INJECTION; OPHTHALMIC; ORAL
Osteomyelitis; Endophthalmitis; Escherichia coli Infections; HIV Infections; Kidney Diseases; Urinary Bladder, Overactive; Appendicitis; Cellulitis; Diabetic Foot; Lymphoma, Non-Hodgkin; Neoplasms; Sarcoidosis; Tuberculosis, Multidrug-Resistant; Cataract; Cystic Fibrosis; Dyspepsia; Endocarditis; Fever; Helicobacter Infections; Hot Flashes; Maxillary Sinusitis; Neutropenia; Otitis Media; Pelvic Inflammatory Disease; Pneumonia, Bacterial; Prostatic Hyperplasia; Prostatitis; Pulmonary Disease, Chronic Obstructive; Pyelonephritis; Skin Diseases; Staphylococcal Infections; Tuberculosis; Acne Vulgaris; Bacterial Infections; Bronchitis, Chronic; Conjunctivitis, Bacterial; Corneal Ulcer; Eye Infections; Infections; Otitis Externa; Pneumonia; Sinusitis; Urinary Tract Infections
DNA gyrase inhibitor
Small molecule
Approved
Unknown
ORAL
Hepatitis C, Chronic; Infertility, Male; Hepatitis C; Hyperoxaluria, Primary; Non-alcoholic Fatty Liver Disease; Obesity; Depressive Disorder; Homocystinuria
Betaine-homocysteine S-methyltransferase substrate
Small molecule
Approved
Unknown
Unknown
Carcinoma, Non-Small-Cell Lung; Dermatitis, Atopic; Edema; Gastroesophageal Reflux; Rhinitis, Allergic, Perennial; Asthma; Rhinitis, Allergic, Seasonal; Hypersensitivity
Unknown
Small molecule
Unknown
Unknown
Unknown
Amyotrophic Lateral Sclerosis; Cystic Fibrosis; Lymphoma; Muscular Atrophy, Spinal; Myelodysplastic-Myeloproliferative Diseases; Myelodysplastic Syndromes; Pyruvate Dehydrogenase Complex Deficiency Disease; Argininosuccinic Aciduria; HIV Infections; Huntington Disease; Leukemia; Machado-Joseph Disease; Tuberculosis, Pulmonary; Hyperammonemia; Urea Cycle Disorders, Inborn
Glutamine sequestering agent
Small molecule
Unknown
Unknown
Unknown
Acquired Immunodeficiency Syndrome; Infections; Tuberculosis; HIV Infections; Virus Diseases
Human immunodeficiency virus type 1 reverse transcriptase inhibitor
Small molecule
Approved
Unknown
Unknown
Sarcoma, Kaposi; Acquired Immunodeficiency Syndrome; HIV Infections; Virus Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Hepatopulmonary Syndrome; Hypotension, Orthostatic; Ischemic Stroke; Ascites; Hypotension; Shock, Septic; Spinal Cord Injuries; Cardiovascular Diseases
Unknown
Enzyme
Approved
Unknown
Unknown
Hypoglycemia; Pancreatic Neoplasms; Pancreatitis; Cystic Fibrosis; Exocrine Pancreatic Insufficiency; Pancreatitis, Chronic
Fatty acids hydrolytic enzyme