Display Options:
Total: 10647
Small molecule
Approved
OTHER
ORAL
Carcinoma, Non-Small-Cell Lung; Insulin Resistance; Malaria; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Acquired Immunodeficiency Syndrome; Pneumonia, Pneumocystis; Severe Acute Respiratory Syndrome; HIV Infections; Infections
Cytochrome P450 3A inhibitor
Unknown
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Pulmonary Disease, Chronic Obstructive
Unknown
Small molecule
Approved
CANCER; OTHER; UROLOGY AND KIDNEY
ORAL
Blast Crisis; Breast Neoplasms; Carcinoma; Endometriosis; Gliosarcoma; Mesothelioma; Stomach Neoplasms; Adrenal Cortex Neoplasms; Biliary Tract Neoplasms; Carcinoid Tumor; Carcinoma, Adenoid Cystic; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Colorectal Neoplasms; Endometrial Neoplasms; Gastrointestinal Stromal Tumors; Glioblastoma; Leukemia, Myeloid, Acute; Melanoma; Myelodysplastic Syndromes; Nasopharyngeal Neoplasms; Pancreatic Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Salivary Gland Neoplasms; Sarcoma; Sarcoma, Alveolar Soft Part; Skin Neoplasms; Solitary Fibrous Tumors; Thyroid Neoplasms; Carcinoma, Pancreatic Ductal; Kidney Neoplasms; Carcinoma, Renal Cell; Neoplasms
Vascular endothelial growth factor receptor inhibitor
Small molecule
Approved
Unknown
Unknown
Asthma; Bronchitis, Chronic; Emphysema; Pulmonary Disease, Chronic Obstructive
Beta-2 adrenergic receptor agonist
Small molecule
Approved
IMMUNE SYSTEM; MUSCULOSKELETAL; OTHER
ORAL
Gliosarcoma; Leukemia, Lymphocytic, Chronic, B-Cell; Arthritis, Psoriatic; Arthritis, Rheumatoid; Cerebral Hemorrhage; Ischemic Stroke; Lymphoma, T-Cell, Cutaneous; Severe Acute Respiratory Syndrome; Sleep Apnea, Obstructive; Multiple Sclerosis, Chronic Progressive; Multiple Sclerosis, Relapsing-Remitting; Psoriasis; Immune System Diseases; Multiple Sclerosis
Kelch-like ECH-associated protein 1 inhibitor
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease
Unknown
Protein
Approved
Unknown
Unknown
Melanoma; Endometrial Neoplasms; Colorectal Neoplasms, Hereditary Nonpolyposis; Epilepsy; Breast Neoplasms; Carcinoma, Squamous Cell
Unknown
Small molecule
Approved
Unknown
Unknown
Brain Neoplasms; Glioma; Kidney Diseases; Liver Diseases; Multiple Myeloma; Adenocarcinoma, Follicular; Ameloblastoma; Carcinoma; Carcinoma, Non-Small-Cell Lung; Erdheim-Chester Disease; Lung Neoplasms; Melanoma; Thyroid Neoplasms; Neoplasms
Unknown
Small molecule
Approved
OTHER
ORAL
Depressive Disorder, Major
Norepinephrine transporter inhibitor
Small molecule
Approved
Unknown
Unknown
Diabetes Mellitus, Type 2; Eye Diseases; Dermatitis; Heart Diseases; Dry Eye Syndromes; Low Back Pain; Lupus Erythematosus, Systemic; Neonatal Sepsis; Obesity; Osteoarthritis, Knee; Periodontal Diseases; Psoriasis; Sarcopenia; Hypertriglyceridemia
Unknown
Unknown
Approved
OTHER
ORAL
Hyperphosphatemia; Renal Insufficiency, Chronic
Phosphate sequestering agent
Unknown
Unknown
Unknown
Unknown
Fatigue Syndrome, Chronic; Pulmonary Disease, Chronic Obstructive; Genital Neoplasms, Female; Heart Failure; Hip Fractures; Inflammatory Breast Neoplasms; Restless Legs Syndrome; Anemia; Anemia, Iron-Deficiency
Supplement
Small molecule
Approved
Unknown
Unknown
Tobacco Use Disorder; Depressive Disorder, Major
Unknown
Oligonucleotide
Approved
Unknown
Unknown
Cardiovascular Diseases
Unknown
Small molecule
Unknown
Unknown
Unknown
Neoplasms; Erdheim-Chester Disease; Multiple Myeloma; Lung Neoplasms; Melanoma; Thyroid Neoplasms
Dual specificity mitogen-activated protein kinase kinase 1 inhibitor
Small molecule
Approved
Unknown
Unknown
Diabetes Mellitus, Type 2; Diabetes Mellitus
Unknown
Unknown
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Asthma; Hyperhidrosis; Pulmonary Disease, Chronic Obstructive
Unknown
Small molecule
Approved
PREGNANCY AND GYNECOLOGY
ORAL
Paget Disease, Extramammary; Atrophy; Dyspareunia; Menopause
Estrogen receptor modulator
Small molecule
Approved
Unknown
ORAL
Amyotrophic Lateral Sclerosis; Acquired Immunodeficiency Syndrome; HIV Infections; Infections; Virus Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Prostatic Neoplasms, Castration-Resistant; Sarcoma; Breast Neoplasms
Unknown
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Cognitive Dysfunction
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Hypospadias; Obesity, Morbid; Pain; Burns; Headache; Postoperative Nausea and Vomiting; Glaucoma
Unknown
Small molecule
Approved
CARDIOVASCULAR; OTHER; RESPIRATORY
ORAL
HIV Infections; Anemia, Sickle Cell; Coronary Disease; Cystic Fibrosis; Raynaud Disease; Scleroderma, Localized; Scleroderma, Systemic; Ulcer; Familial Primary Pulmonary Hypertension; Hypertension; Hypertension, Pulmonary
Soluble guanylate cyclase positive allosteric modulator
Small molecule
Approved
Unknown
Unknown
Renal Insufficiency, Chronic; Hepatitis C; Hepatitis C, Chronic; Virus Diseases
Unknown
Small molecule
Approved
CANCER; HEMATOLOGY; OTHER
ORAL
Amyloidosis; Anemia, Sickle Cell; Castleman Disease; Hodgkin Disease; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Neoplasms; Pancreatic Neoplasms; Small Cell Lung Carcinoma; Waldenstrom Macroglobulinemia; Amyloidosis, Familial; Graft vs Host Disease; Leukemia, Plasma Cell; Lung Diseases, Interstitial; Medulloblastoma; Myeloproliferative Disorders; Plasmacytoma; Polycythemia Vera; Prostatic Neoplasms, Castration-Resistant; Pulmonary Fibrosis; Sarcoma; Sarcoma, Kaposi; Scleroderma, Systemic; Telangiectasia, Hereditary Hemorrhagic; Primary Myelofibrosis; Immune System Diseases; Multiple Myeloma
CRL4(CRBN) E3 ubiquitin ligase inhibitor
Small molecule
Approved
Unknown
ORAL
Liver Diseases; Attention Deficit Disorder with Hyperactivity; Bipolar Disorder; Feeding and Eating Disorders; Anxiety Disorders; Depressive Disorder, Major; Depressive Disorder
Unknown
Small molecule
Approved
Unknown
Unknown
Asthma; Pulmonary Disease, Chronic Obstructive
Unknown
Antibody
Approved
CANCER
INJECTION
Burkitt Lymphoma; Colorectal Neoplasms; Hodgkin Disease; Leukemia; Leukemia, Prolymphocytic; Mycosis Fungoides; Renal Insufficiency, Chronic; Carcinoma, Non-Small-Cell Lung; Graft vs Host Disease; Leukemia, Hairy Cell; Lymphoma; Lymphoma, Mantle-Cell; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Waldenstrom Macroglobulinemia; Kidney Diseases; Lupus Erythematosus, Systemic; Lupus Nephritis; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, Follicular; Neoplasms
B-lymphocyte antigen CD20 binding agent
Small molecule
Approved
HEMATOLOGY
ORAL
Breast Neoplasms; Carcinoma, Renal Cell; Colonic Neoplasms; Colorectal Neoplasms; Glioblastoma; Hematologic Neoplasms; Leukemia, Lymphoid; Liver Diseases; Lung Neoplasms; Myelodysplastic Syndromes; Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms, Castration-Resistant; Amyloidosis; Anemia, Hemolytic, Autoimmune; Burkitt Lymphoma; Carcinoid Tumor; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Esophageal Neoplasms; Food Hypersensitivity; Hodgkin Disease; Leukemia; Leukemia, Hairy Cell; Leukemia, Mast-Cell; Leukemia, Myeloid, Acute; Leukemia, Prolymphocytic; Leukemia, Prolymphocytic, T-Cell; Lymphoma, B-Cell, Marginal Zone; Melanoma; Multiple Myeloma; Severe Acute Respiratory Syndrome; Graft vs Host Disease; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, Mantle-Cell; Waldenstrom Macroglobulinemia
Tyrosine-protein kinase BTK inhibitor
Antibody
Approved
Unknown
Unknown
Carcinoma, Non-Small-Cell Lung; Multiple Myeloma; Neoplasm Metastasis; Ovarian Neoplasms; Salivary Gland Neoplasms; Stomach Neoplasms; Breast Neoplasms; Neoplasms
Receptor protein-tyrosine kinase erbB-2 inhibitor
Unknown
Approved
Unknown
Unknown
Unknown
Unknown