Display Options:
Total: 6532
Small molecule
Investigational
Unknown
Unknown
Neoplasms; Prostatic Neoplasms
Tyrosine-protein kinase TIE-2 inhibitor
Small molecule
Investigational
Unknown
Unknown
Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Neoplasms; Carcinoma, Squamous Cell
PI3-kinase p110-delta subunit inhibitor
Small molecule
Investigational
Unknown
Unknown
Unknown
Calcium-activated potassium channel subunit alpha-1 activator
Small molecule
Investigational
Unknown
Unknown
Leukemia, Myeloid, Acute; Neoplasms; Paraganglioma
Isocitrate dehydrogenase [NADP] cytoplasmic inhibitor
Small molecule
Investigational
Unknown
Unknown
Irritable Bowel Syndrome; Schizophrenia
Neurokinin 3 receptor antagonist
Small molecule
Investigational
Unknown
Unknown
Melanoma; Prostatic Neoplasms, Castration-Resistant; Skin Aging; Aging; Breast Neoplasms; Child Development Disorders, Pervasive; Depressive Disorder; Diabetes Mellitus, Type 2; Kidney Diseases; Lung Neoplasms; Parkinson Disease; Prostatic Neoplasms; Renal Insufficiency, Chronic; Schizophrenia; Subarachnoid Hemorrhage; Urinary Bladder Neoplasms; Autistic Disorder; Psychotic Disorders
Unknown
Small molecule
Investigational
Unknown
Unknown
Colorectal Neoplasms
Unknown
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
Small molecule
Investigational
Unknown
Unknown
Renal Insufficiency, Chronic; Coronary Disease; Erectile Dysfunction
Rho-associated protein kinase inhibitor
Small molecule
Investigational
Unknown
Unknown
Osteoporosis
Unknown
Small molecule
Investigational
Unknown
Unknown
Diabetes Mellitus, Type 2
Unknown
Small molecule
Investigational
Unknown
Unknown
Neoplasms
Tyrosine-protein kinase JAK2 inhibitor
Small molecule
Investigational
Unknown
Unknown
Candidiasis; Eczema; Gingivitis; Tinea Pedis
Unknown
Small molecule
Investigational
Unknown
Unknown
Neoplasms; Sarcoma, Kaposi
Unknown
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
Small molecule
Investigational
Unknown
Unknown
Infertility; Asthma; Chronic Urticaria; Pulmonary Disease, Chronic Obstructive
G protein-coupled receptor 44 antagonist
Small molecule
Investigational
Unknown
Unknown
Acne Vulgaris
Acetyl-CoA carboxylase inhibitor
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
Small molecule
Investigational
Unknown
Unknown
Carcinoma, Non-Small-Cell Lung; Colonic Neoplasms; Mesothelioma; Rectal Neoplasms
Tubulin inhibitor
Small molecule
Investigational
Unknown
Unknown
Colorectal Neoplasms; Neoplasms; Head and Neck Neoplasms
Thymidylate synthase inhibitor
Small molecule
Investigational
Unknown
Unknown
Alzheimer Disease
GABA-A receptor; anion channel inverse agonist
Small molecule
Investigational
Unknown
Unknown
Infections
Unknown
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
Small molecule
Investigational
Unknown
Unknown
Coronary Disease
Unknown
Small molecule
Investigational
Unknown
Unknown
Diabetes Mellitus, Type 2; Multiple Sclerosis, Relapsing-Remitting
Peroxisome proliferator-activated receptor gamma modulator
Small molecule
Investigational
Unknown
Unknown
HIV Infections
Unknown
Small molecule
Investigational
Unknown
Unknown
Sleep Initiation and Maintenance Disorders; Sleep Wake Disorders
Orexin receptor 1 antagonist
Small molecule
Investigational
Unknown
Unknown
Arthritis, Rheumatoid; Multiple Sclerosis, Relapsing-Remitting
C-C chemokine receptor type 2 antagonist
Small molecule
Investigational
Unknown
Unknown
Lymphoma; Endometrial Neoplasms; Uterine Cervical Neoplasms
DNA disrupting agent
Small molecule
Investigational
Unknown
Unknown
Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Precursor Cell Lymphoblastic Leukemia-Lymphoma
Tyrosine-protein kinase ABL inhibitor
Small molecule
Investigational
Unknown
Unknown
Fuchs' Endothelial Dystrophy
Rho-associated protein kinase inhibitor
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
Small molecule
Investigational
Unknown
Unknown
Alzheimer Disease
Muscarinic acetylcholine receptor M1 positive allosteric modulator
Small molecule
Investigational
Unknown
Unknown
Alcoholism; Obesity; Sexual Dysfunction, Physiological
Mu opioid receptor antagonist
Small molecule
Investigational
Unknown
Unknown
Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Carcinoma, Pancreatic Ductal; Leukemia, Myeloid, Acute; Lymphoma, Large B-Cell, Diffuse; Prostatic Neoplasms, Castration-Resistant; Glioblastoma
Bromodomain and extra-terminal motif (BET) inhibitor