Display Options:
Total: 6532
Small molecule
Approved
OTHER
ORAL
Breast Neoplasms; Hypogonadism; Neoplasms; Orchitis
Androgen Receptor agonist
Small molecule
Approved
Unknown
Unknown
Dementia; Depressive Disorder; Schizophrenia; Anxiety
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Hypertension
Synaptic vesicular amine transporter inhibitor
Small molecule
Approved
Unknown
Unknown
Digestive System Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Radiopharmaceutical
Small molecule
Approved
OTHER
ORAL
Unknown
Bacterial 70S ribosome inhibitor
Small molecule
Approved
OTHER
ORAL
Hypertension
Synaptic vesicular amine transporter inhibitor
Small molecule
Approved
OTHER
ORAL
Psychotic Disorders
Dopamine D2 receptor antagonist
Small molecule
Approved
OTHER
ORAL
Carcinoma, Pancreatic Ductal; Lymphoma, Mantle-Cell; Glomerulonephritis, Membranous; Glomerulosclerosis, Focal Segmental; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma; Lymphoma, B-Cell, Marginal Zone; Stomach Neoplasms; Hodgkin Disease; Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Atherosclerosis; Chemical and Drug Induced Liver Injury; Cognitive Dysfunction; DiGeorge Syndrome; Friedreich Ataxia; Frontotemporal Dementia; Gangliosidoses; Gaucher Disease; Hearing Loss, Noise-Induced; Hyperuricemia; Immune System Diseases; Intussusception; Lymphoma, Follicular; Mucocutaneous Lymph Node Syndrome; Muscular Diseases; Myasthenia Gravis; Optic Nerve Diseases; Ovarian Hyperstimulation Syndrome; Parkinson Disease; Radius Fractures; Shoulder Pain; Stiff-Person Syndrome; Adenomatous Polyposis Coli; Amyotrophic Lateral Sclerosis; Anemia, Aplastic; Appendicitis; Blastic Plasmacytoid Dendritic Cell Neoplasm; Breast Neoplasms; Bronchiolitis Obliterans Syndrome; Burkitt Lymphoma; Carcinoma, Non-Small-Cell Lung; Coronavirus Infections; Death, Sudden, Cardiac; Fallopian Tube Neoplasms; Fanconi Anemia; Fasciitis, Plantar; Graves Ophthalmopathy; Hantavirus Infections; Hepatitis, Alcoholic; Hyperlipoproteinemia Type I; IgA Vasculitis; Immunoblastic Lymphadenopathy; Immunoglobulin G4-Related Disease; Kidney Failure, Chronic; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, AIDS-Related; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Lymphoproliferative Disorders; Melanoma; Migraine Disorders; Myelodysplastic-Myeloproliferative Diseases; Myelodysplastic Syndromes; Myeloproliferative Disorders; Nasal Polyps; Neoplasms; Neoplasms, Plasma Cell; Neuromyelitis Optica; Osteoarthritis, Knee; Ovarian Neoplasms; Prostatic Neoplasms; Purpura, Thrombotic Thrombocytopenic; Radiculopathy; Sinusitis; Spasms, Infantile; Spondylarthropathies; Spondylitis, Ankylosing; Abdominal Pain; Aging; Anti-Neutrophil Cytoplasmic Antibody-Associated Vasculitis; Bell Palsy; Bronchopulmonary Dysplasia; Carpal Tunnel Syndrome; Colitis; Deglutition Disorders; Dermatomyositis; Edema; Erythema Multiforme; Glomerulonephritis, IGA; Glomerulonephritis, Membranous; Graft vs Host Disease; Granulomatosis with Polyangiitis; Heart Arrest; Heart Diseases; Hematologic Neoplasms; Hematoma, Subdural, Intracranial; Hodgkin Disease; Idiopathic Pulmonary Fibrosis; Ischemic Stroke; Kidney Diseases; Language Disorders; Leukemia; Leukemia, Biphenotypic, Acute; Lupus Erythematosus, Systemic; Lupus Nephritis; Lymphohistiocytosis, Hemophagocytic; Lymphoma; Macrophage Activation Syndrome; Meniere Disease; Microscopic Polyangiitis; Multiple Myeloma; Multiple Sclerosis, Chronic Progressive; Multiple Sclerosis, Relapsing-Remitting; Myocarditis; Optic Neuritis; Optic Neuropathy, Ischemic; Pain; Pneumonia, Pneumocystis; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms, Castration-Resistant; Pulmonary Disease, Chronic Obstructive; Pulpitis; Purpura, Thrombocytopenic, Idiopathic; Renal Insufficiency; Renal Insufficiency, Chronic; Respiratory Distress Syndrome; Respiratory Tract Diseases; Scleroderma, Systemic; Severe Acute Respiratory Syndrome; Specific Language Disorder; Spinal Cord Injuries; Stroke; Thrombocytopenia; Urinary Tract Infections; Vestibular Neuronitis; Wounds and Injuries; Acne Vulgaris; Arthritis, Juvenile; Arthritis, Psoriatic; Arthritis, Rheumatoid; Asthma; Bursitis; Colitis, Ulcerative; Crohn Disease; Dermatitis, Atopic; Endocrine System Diseases; Inflammation; Multiple Sclerosis; Osteoarthritis; Pneumonia; Tenosynovitis; Uveitis, Posterior
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Carcinoma, Hepatocellular; Motion Sickness; Smoking Cessation; Vertigo; Hypersensitivity
Unknown
Small molecule
Approved
Unknown
Unknown
Hypersensitivity
Unknown
Small molecule
Approved
OTHER
ORAL
Unknown
Muscarinic acetylcholine receptor M1 antagonist
Small molecule
Approved
OTHER
ORAL
Epilepsy; Seizures
Sodium channel alpha subunit blocker
Small molecule
Approved
Unknown
Unknown
Low Back Pain
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Common Cold; Cough; Hypersensitivity; Nasal Obstruction; Rhinitis, Allergic, Seasonal; Sinusitis
Histamine H1 receptor antagonist
Small molecule
Approved
OTHER
RECTAL
Colonic Neoplasms; Delirium; Glioblastoma; Neonatal Abstinence Syndrome; Severe Acute Respiratory Syndrome; Conduct Disorder; Porphyrias; Postoperative Nausea and Vomiting; Psychotic Disorders; Schizophrenia
D2-like dopamine receptor antagonist
Small molecule
Approved
Unknown
Unknown
Digestive System Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Pain
Unknown
Small molecule
Approved
OTHER
ORAL
Epilepsy; Seizures
Voltage-gated T-type calcium channel blocker
Small molecule
Approved
OTHER
IM-IV; INJECTION; ORAL
Liver Cirrhosis; Pain
Carbonic anhydrase I inhibitor
Small molecule
Approved
OTHER
ORAL
Diabetic Retinopathy; Macular Degeneration; Nasal Polyps; Neuralgia; Optic Neuropathy, Ischemic; Rotator Cuff Injuries; Sinusitis; Abdominal Pain; Acneiform Eruptions; Alopecia Areata; Dermatitis, Atopic; Geographic Atrophy; Lichen Planus, Oral; Melanoma; Melanosis; Osteoarthritis, Knee; Psoriasis; Shoulder Pain; Vascular Diseases; Vitiligo; Wet Macular Degeneration; Corneal Edema; Keloid; Lung Diseases; Macular Edema; Orbital Pseudotumor; Osteoarthritis; Osteoarthritis, Hip; Pain; Pancreatitis, Chronic; Pulmonary Disease, Chronic Obstructive; Radiculopathy; Retinal Vein Occlusion; Rhinitis, Allergic, Perennial; Rhinitis, Allergic, Seasonal; Eye Diseases; Hemorrhoids; Lung Diseases, Obstructive; Nasal Obstruction; Skin Diseases
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
ORAL
Unknown
Vitamin K-dependent gamma-carboxylase inhibitor
Small molecule
Approved
OTHER
OPHTHALMIC
Glaucoma
Acetylcholinesterase inhibitor
Small molecule
Approved
OTHER
ORAL
Melanoma; Venous Thrombosis; Thrombosis
Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor
Small molecule
Approved
OTHER
INJECTION; ORAL
Cocaine-Related Disorders; Ischemic Stroke; Anxiety; Dementia; Depressive Disorder; Psychomotor Agitation; Postoperative Nausea and Vomiting; Psychotic Disorders; Schizophrenia
Dopamine D2 receptor antagonist
Small molecule
Approved
OTHER
ORAL
Diabetes Mellitus; Diabetes Mellitus, Type 2
Sulfonylurea receptor 1, Kir6.2 blocker
Small molecule
Approved
OTHER
ORAL
Unknown
Intermediate conductance calcium-activated potassium channel protein 4 opener
Small molecule
Approved
Unknown
Unknown
Unknown
Alpha-1a adrenergic receptor agonist
Small molecule
Approved
OTHER
ORAL
Cough
Slowly adapting pulmonary stretch receptor inhibitor
Small molecule
Approved
OTHER
ORAL
Atherosclerosis; Coronary Disease; Diabetes Mellitus, Type 2; Heart Diseases; Hypercholesterolemia; Cardiovascular Diseases; Edema; Glomerulonephritis; Heart Failure; Hypertension; Kidney Failure, Chronic; Nephrotic Syndrome; Toxemia
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
EYE; OTHER
INTRAOCULAR; INTRAVITREAL; OPHTHALMIC; ORAL; TOPICAL
Adrenal Insufficiency; Alcoholism; Anaphylaxis; Aortic Coarctation; Brain Edema; Croup; Esophageal Neoplasms; Glioblastoma; Graves Disease; Head and Neck Neoplasms; Hypertension; Hyperuricemia; Ileus; Keratoconus; Lacrimal Apparatus Diseases; Leukemia, Hairy Cell; Lymphoma, T-Cell, Cutaneous; Meningeal Carcinomatosis; Osteoarthritis, Knee; Pulpitis; Radius Fractures; Retinopathy of Prematurity; Rhabdomyolysis; Rheumatic Diseases; Scleritis; Sepsis; Sinusitis; Tooth Diseases; Vestibular Neuronitis; Vitiligo; Appendicitis; Blast Crisis; Blastic Plasmacytoid Dendritic Cell Neoplasm; Brain Neoplasms; Breast Carcinoma In Situ; Bronchiolitis Obliterans Syndrome; Burkitt Lymphoma; Carcinoma, Renal Cell; Carcinoma, Squamous Cell; Castleman Disease; Cholangiocarcinoma; Choroidal Neovascularization; Dry Eye Syndromes; Dyspnea; Endocrine Gland Neoplasms; Endometrial Neoplasms; Fasciitis, Plantar; Glomerulonephritis; Gout; Hearing Loss; Hearing Loss, Sensorineural; Heart Failure; Hematologic Neoplasms; Hematoma, Subdural, Intracranial; Hemorrhage; Histiocytosis, Langerhans-Cell; Histiocytosis, Sinus; Hypocalcemia; IgA Vasculitis; Immune System Diseases; Intestinal Obstruction; Intracranial Hypertension; Lassa Fever; Leptospirosis; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Plasma Cell; Leukemia, T-Cell; Lichen Planus; Liposarcoma, Myxoid; Liver Neoplasms; Lung Diseases, Obstructive; Lung Neoplasms; Lymphoma, Large-Cell, Anaplastic; Lymphoma, T-Cell, Peripheral; Macular Degeneration; Melanoma; Meningitis; Meningitis, Cryptococcal; Mesothelioma; Mouth Neoplasms; Nasopharyngeal Carcinoma; Neck Pain; Neoplasm Metastasis; Nervous System Diseases; Paget Disease, Extramammary; Pancreatic Neoplasms; Papilledema; Pharyngitis; POEMS Syndrome; Premature Birth; Pulmonary Fibrosis; Purpura, Thrombotic Thrombocytopenic; Radiculopathy; Rectal Neoplasms; Red-Cell Aplasia, Pure; Retinal Vein Occlusion; Stomach Neoplasms; Tonsillitis; Toxoplasmosis, Cerebral; Tuberculosis; Urinary Bladder Neoplasms; Uveitis, Intermediate; Wet Macular Degeneration; Xerostomia; Amyloidosis; Amyloidosis, Familial; Anemia; Anemia, Refractory; Anemia, Refractory, with Excess of Blasts; Anemia, Sickle Cell; Atrioventricular Block; Back Pain; Blepharitis; Breast Neoplasms; Bronchiolitis; Bronchopulmonary Dysplasia; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Cataract; Chronic Pain; Colorectal Neoplasms; Conjunctivitis, Viral; Corneal Edema; Cysticercosis; Deafness; Deglutition Disorders; Encephalitis, Herpes Simplex; Fatigue; Genital Neoplasms, Female; Genital Neoplasms, Male; Glaucoma; Glomerulosclerosis, Focal Segmental; Graft vs Host Disease; Granuloma, Lethal Midline; Headache; HELLP Syndrome; Hernias, Diaphragmatic, Congenital; Hodgkin Disease; Hypersensitivity; Immunoglobulin Light-chain Amyloidosis; Influenza, Human; Kidney Failure, Chronic; Knee Injuries; Leiomyoma; Leukemia, Biphenotypic, Acute; Leukemia, Erythroblastic, Acute; Leukemia, Lymphoid; Leukemia, Megakaryoblastic, Acute; Leukemia, Monocytic, Acute; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Acute; Leukemia, Myelomonocytic, Chronic; Lichen Planus, Oral; Liver Cirrhosis; Lymphohistiocytosis, Hemophagocytic; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Malaria; Mastoiditis; Meniere Disease; Migraine Disorders; Multiple Myeloma; Multiple Sclerosis, Chronic Progressive; Myelodysplastic Syndromes; Nausea; Neoplasms, Plasma Cell; Nephrosis; Neuralgia; Otitis Externa; Otitis Media; Ovarian Hyperstimulation Syndrome; Ovarian Neoplasms; Pain; Pelvic Organ Prolapse; Plasmacytoma; Pneumonia, Viral; Postoperative Complications; Postoperative Nausea and Vomiting; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Pregnancy; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Renal Insufficiency, Chronic; Respiratory Distress Syndrome; Respiratory Insufficiency; Rhinitis, Allergic, Perennial; Rotator Cuff Injuries; Sarcoma; Sciatica; Severe Acute Respiratory Syndrome; Sleep Apnea, Obstructive; Small Cell Lung Carcinoma; Smoldering Multiple Myeloma; Specific Language Disorder; Strabismus; Subarachnoid Hemorrhage; Urinary Tract Infections; Uveitis, Anterior; Vaginosis, Bacterial; Vitreoretinopathy, Proliferative; Vomiting; Waldenstrom Macroglobulinemia; Wounds and Injuries; Wrist Fractures; Acne Vulgaris; Addison Disease; Adrenal Hyperplasia, Congenital; Adrenocortical Hyperfunction; Anemia, Aplastic; Anemia, Hemolytic; Arthritis, Gouty; Arthritis, Juvenile; Arthritis, Psoriatic; Arthritis, Rheumatoid; Asthma; Bursitis; Chorioretinitis; Choroiditis; Colitis, Ulcerative; Conjunctivitis, Allergic; Corneal Injuries; Crohn Disease; Dermatitis; Dermatitis, Atopic; Dermatitis, Contact; Dermatitis, Exfoliative; Dermatitis Herpetiformis; Dermatitis, Seborrheic; Diabetic Retinopathy; Erythema Multiforme; Eye Diseases; Hemorrhoids; Herpes Simplex; Herpes Zoster Ophthalmicus; Hypercalcemia; Infections; Inflammation; Iridocyclitis; Iritis; Keratitis; Leukemia; Lupus Erythematosus, Systemic; Lymphoma; Macular Edema; Multiple Sclerosis; Mycosis Fungoides; Myocarditis; Nasal Obstruction; Neoplasms; Nephrotic Syndrome; Ophthalmia, Sympathetic; Optic Neuritis; Osteoarthritis; Pemphigus; Peptic Ulcer; Pneumonia; Psoriasis; Pulmonary Eosinophilia; Purpura, Thrombocytopenic, Idiopathic; Rhinitis, Allergic; Rhinitis, Allergic, Seasonal; Sarcoidosis; Serum Sickness; Spondylitis, Ankylosing; Stevens-Johnson Syndrome; Synovitis; Tennis Elbow; Tenosynovitis; Thrombocytopenia; Thyroiditis, Subacute; Trichinellosis; Tuberculosis, Meningeal; Tuberculosis, Pulmonary; Uveitis; Uveitis, Posterior
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
ORAL
Unknown
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
ORAL
Hypokalemic Periodic Paralysis; Myotonic Disorders; Paralysis, Hyperkalemic Periodic; Glaucoma
Carbonic anhydrase II inhibitor