Display Options:
Total: 6532
Small molecule
Approved
OTHER
ORAL
Atherosclerosis; Coronary Disease; Diabetes Mellitus, Type 2; Heart Diseases; Hypercholesterolemia; Cardiovascular Diseases; Edema; Glomerulonephritis; Heart Failure; Hypertension; Kidney Failure, Chronic; Nephrotic Syndrome; Toxemia
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
OTHER
ORAL
Unknown
DNA inhibitor
Small molecule
Approved
OTHER
ORAL
Unknown
Bacterial penicillin-binding protein inhibitor
Small molecule
Approved
OTHER
ORAL
Hypokalemic Periodic Paralysis; Myotonic Disorders; Paralysis, Hyperkalemic Periodic; Glaucoma
Carbonic anhydrase II inhibitor
Small molecule
Approved
OTHER
ORAL
Low Back Pain; Pain; Spasm
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL
Adenocarcinoma of Lung; Anemia; Biliary Tract Neoplasms; Breast Carcinoma In Situ; Carcinoma, Medullary; Carcinoma, Pancreatic Ductal; Chordoma; Desmoplastic Small Round Cell Tumor; Fibroma; Fibrosarcoma; Glioblastoma; Glomerulosclerosis, Focal Segmental; Hepatoblastoma; Histiocytoma; HIV Infections; Leukemia, Myeloid; Leukemia, Plasma Cell; Liposarcoma; Liposarcoma, Myxoid; Lymphoma, Primary Effusion; Muscular Diseases; Myasthenia Gravis; Mycosis Fungoides; Myoepithelioma; Nasopharyngeal Carcinoma; Nasopharyngeal Neoplasms; Nausea; Neoplasm Metastasis; Osteogenesis Imperfecta; Renal Insufficiency; Sarcoma, Clear Cell; Sarcoma, Synovial; Sezary Syndrome; Stiff-Person Syndrome; Urinary Bladder Neoplasms; Acquired Immunodeficiency Syndrome; Adrenoleukodystrophy; Anemia, Sickle Cell; Arthritis, Rheumatoid; Blast Crisis; Blastic Plasmacytoid Dendritic Cell Neoplasm; Breast Neoplasms, Male; Bronchiolitis Obliterans Syndrome; Carcinoma, Merkel Cell; Castleman Disease; Colorectal Neoplasms; Crohn Disease; Endometrial Neoplasms; Epidermolysis Bullosa; Esophageal Neoplasms; Esthesioneuroblastoma, Olfactory; Fanconi Anemia; Fucosidosis; Gangliosidosis, GM1; Gaucher Disease; Glioma; Gliosarcoma; Granulomatous Disease, Chronic; Head and Neck Neoplasms; Hematologic Diseases; Hereditary Breast and Ovarian Cancer Syndrome; Histiocytosis, Langerhans-Cell; IgA Vasculitis; Immune System Diseases; Immunoglobulin Light-chain Amyloidosis; Immunologic Deficiency Syndromes; Kidney Failure, Chronic; Leukemia, Myelomonocytic, Juvenile; Leukemia, Prolymphocytic; Leukodystrophy, Globoid Cell; Leukodystrophy, Metachromatic; Liver Neoplasms; Lupus Erythematosus, Systemic; Lymphohistiocytosis, Hemophagocytic; Lymphoma, AIDS-Related; Lymphoma, B-Cell; Lymphoma, Large-Cell, Anaplastic; Lymphoma, T-Cell; Lymphoproliferative Disorders; Mesothelioma; Mouth Neoplasms; Myelodysplastic-Myeloproliferative Diseases; Neuroectodermal Tumors, Primitive, Peripheral; Neuroendocrine Tumors; Neuromyelitis Optica; Neuronal Ceroid-Lipofuscinoses; Niemann-Pick Diseases; Osteopetrosis; Osteosarcoma; Pancreatic Neoplasms; Paraganglioma; Peritoneal Neoplasms; Plasmacytoma; Polyradiculoneuropathy, Chronic Inflammatory Demyelinating; Primary Immunodeficiency Diseases; Primary Myelofibrosis; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Purpura, Thrombocytopenic, Idiopathic; Rectal Neoplasms; Sandhoff Disease; Sarcoidosis; Skin Neoplasms; Squamous Intraepithelial Lesions; Takayasu Arteritis; Tay-Sachs Disease; Thalassemia; Thymoma; Thyroid Neoplasms; Tuberculosis; Uterine Cervical Neoplasms; Uveal Melanoma; Vasculitis; Wolman Disease; Adenocarcinoma; Amyloidosis; Amyloidosis, Familial; Anemia, Aplastic; Anemia, Refractory; Anemia, Refractory, with Excess of Blasts; Anti-Neutrophil Cytoplasmic Antibody-Associated Vasculitis; Attention Deficit Disorder with Hyperactivity; Behcet Syndrome; Bone Marrow Failure Disorders; Brain Neoplasms; Burkitt Lymphoma; Carcinoma; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Choroid Plexus Neoplasms; Condylomata Acuminata; Ependymoma; Fallopian Tube Neoplasms; Ganglioneuroblastoma; Gestational Trophoblastic Disease; Glomerulonephritis, IGA; Glomerulonephritis, Membranous; Graft vs Host Disease; Granuloma, Lethal Midline; Granulomatosis with Polyangiitis; Hematologic Neoplasms; Idiopathic Pulmonary Fibrosis; Immunoblastic Lymphadenopathy; Infertility; Inflammatory Breast Neoplasms; Kidney Diseases; Kidney Neoplasms; Leukemia; Leukemia, Biphenotypic, Acute; Leukemia, Erythroblastic, Acute; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Lymphoid; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Megakaryoblastic, Acute; Leukemia, Monocytic, Acute; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Acute; Leukemia, Myelomonocytic, Chronic; Lung Diseases; Lung Neoplasms; Lupus Nephritis; Lymphoma, B-Cell, Marginal Zone; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Lymphoma, T-Cell, Peripheral; Medulloblastoma; Melanoma; Menopause; Microscopic Polyangiitis; Multiple Sclerosis; Multiple Sclerosis, Chronic Progressive; Multiple Sclerosis, Relapsing-Remitting; Myelodysplastic Syndromes; Myeloproliferative Disorders; Neoplasms, Germ Cell and Embryonal; Neoplasms, Plasma Cell; Neuroblastoma; Neuroectodermal Tumors, Primitive; Neutropenia; Ovarian Neoplasms; Pemphigus; Postoperative Nausea and Vomiting; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Pulmonary Fibrosis; Red-Cell Aplasia, Pure; Renal Insufficiency, Chronic; Retinoblastoma; Rhabdomyosarcoma; Rhabdomyosarcoma, Alveolar; Rhabdomyosarcoma, Embryonal; Sarcoma; Sarcoma, Ewing; Scleritis; Scleroderma, Localized; Scleroderma, Systemic; Small Cell Lung Carcinoma; Squamous Cell Carcinoma of Head and Neck; Testicular Neoplasms; Thrombocytopenia; Thrombosis; Triple Negative Breast Neoplasms; Waldenstrom Macroglobulinemia; Wilms Tumor; Breast Neoplasms; Hodgkin Disease; Lymphoma; Multiple Myeloma; Neoplasms; Nephrotic Syndrome
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Schizophrenia; Psychotic Disorders
Unknown
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY
ORAL
Alzheimer Disease; Depression; Depressive Disorder; Depressive Disorder, Major
Monoamine oxidase inhibitor
Small molecule
Approved
OTHER
ORAL
Gout
Solute carrier family 22 member 12 inhibitor
Small molecule
Approved
OTHER
INJECTION; INTRAVENOUS
Anemia; Chordoma; Crohn Disease; Fallopian Tube Neoplasms; Immune System Diseases; Kidney Neoplasms; Liver Neoplasms; Neoplasms, Germ Cell and Embryonal; Neoplasms, Neuroepithelial; Ovarian Neoplasms; Peritoneal Neoplasms; Severe Combined Immunodeficiency; Wiskott-Aldrich Syndrome; Anemia, Sickle Cell; Breast Neoplasms, Male; Glioma; Hematologic Diseases; Hematologic Neoplasms; Inflammatory Breast Neoplasms; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Lymphoma, T-Cell, Peripheral; Multiple Myeloma; Myelodysplastic Syndromes; Myeloproliferative Disorders; Neoplasms, Plasma Cell; Osteosarcoma; Primary Myelofibrosis; Sarcoma; Brain Neoplasms; Breast Neoplasms; Central Nervous System Neoplasms; Ganglioneuroblastoma; Graft vs Host Disease; Leukemia; Medulloblastoma; Neuroblastoma; Neuroectodermal Tumors, Primitive; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Retinoblastoma; Adenocarcinoma; Carcinoma; Hematopoietic Stem Cell Transplantation; Hodgkin Disease; Neoplasms
DNA inhibitor
Small molecule
Approved
Unknown
Unknown
Obesity
Unknown
Small molecule
Approved
Unknown
Unknown
Breast Neoplasms; Dysthymic Disorder; Photosensitivity Disorders; Rosacea; Somatoform Disorders; Anxiety; Chest Pain; Death, Sudden, Cardiac; Dementia; Digestive System Diseases; Gastroesophageal Reflux; Low Back Pain; Myocardial Infarction; Schizophrenia; Urinary Incontinence, Stress; Ventricular Fibrillation; Depressive Disorder
Unknown
Small molecule
Approved
Unknown
Unknown
Bulimia Nervosa; Kidney Diseases; Liver Diseases; Substance-Related Disorders; Diabetes Mellitus; Obesity, Morbid; Obesity
Norepinephrine transporter releasing agent
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Diabetes Mellitus; Lecithin Cholesterol Acyltransferase Deficiency; Metabolic Syndrome; Photosensitivity Disorders; Diabetic Nephropathies; Kidney Diseases; Atherosclerosis; Coronary Disease; Death, Sudden, Cardiac; Diabetes Mellitus, Type 2; Essential Hypertension; Hypercholesterolemia; Kidney Calculi; Polycystic Kidney, Autosomal Dominant; Pre-Eclampsia; Angina Pectoris; Cardiovascular Diseases; Edema; Glomerulonephritis; Heart Failure; Hypertension; Kidney Failure, Chronic; Liver Cirrhosis; Myocardial Infarction; Nephrotic Syndrome; Toxemia
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
Unknown
Unknown
Anxiety; Cocaine-Related Disorders; Dementia; Depressive Disorder; Schizophrenia; Parkinson Disease
Unknown
Small molecule
Approved
OTHER
INJECTION; INTERSTITIAL; INTRAVENOUS
Arthritis, Rheumatoid; Bone Neoplasms; Brain Neoplasms; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Lung Neoplasms; Lymphedema; Melanoma; Neoplasms; Nervous System Neoplasms; Rotator Cuff Injuries; Uterine Cervical Neoplasms; Breast Neoplasms; Head and Neck Neoplasms; Ovarian Neoplasms; Periodontitis; Sarcoma; Wounds and Injuries; Colorectal Neoplasms; Endometrial Neoplasms; Periodontal Diseases; Retinal Perforations; Stomach Neoplasms
Unknown
Small molecule
Approved
OTHER
ORAL
Cardiovascular Diseases; Hypertension
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
Unknown
Unknown
Macular Edema; Scleritis; Cataract; Dry Eye Syndromes; Uveitis, Anterior
Unknown
Small molecule
Approved
Unknown
Unknown
Neuralgia; Chronic Pain; Gout; Optic Neuritis; Shoulder Impingement Syndrome; Tennis Elbow; Carpal Tunnel Syndrome; Low Back Pain; Pain; Anemia; Arthritis, Rheumatoid; Asthma; Brain Neoplasms; Bursitis; Communicable Diseases; Dermatitis; Leukemia; Lymphoma; Nephrotic Syndrome; Osteoarthritis; Serum Sickness; Uveitis
Glucocorticoid receptor agonist
Small molecule
Approved
Unknown
Unknown
Hematologic Neoplasms; Influenza, Human; Multiple Myeloma; Multiple Sclerosis, Relapsing-Remitting; Plasmacytoma; Rotator Cuff Injuries; Severe Acute Respiratory Syndrome; Spinal Stenosis; Ischemia; Peripheral Arterial Disease; Ataxia Telangiectasia; Joint Diseases; Addison Disease; Adrenal Hyperplasia, Congenital; Adrenal Insufficiency; Anemia, Aplastic; Anemia, Hemolytic; Arthritis, Gouty; Arthritis, Juvenile; Arthritis, Psoriatic; Arthritis, Rheumatoid; Asthma; Brain Edema; Bursitis; Chorioretinitis; Choroiditis; Colitis, Ulcerative; Conjunctivitis, Allergic; Crohn Disease; Dermatitis, Atopic; Dermatitis, Contact; Dermatitis, Exfoliative; Dermatitis Herpetiformis; Dermatitis, Seborrheic; Erythema Multiforme; Herpes Simplex; Herpes Zoster Ophthalmicus; Hypercalcemia; Inflammation; Iridocyclitis; Iritis; Keratitis; Laryngeal Edema; Leukemia; Lupus Erythematosus, Systemic; Lymphoma; Mycosis Fungoides; Myocarditis; Nephrotic Syndrome; Ophthalmia, Sympathetic; Optic Neuritis; Osteoarthritis; Pemphigus; Peptic Ulcer; Pneumonia; Psoriasis; Pulmonary Eosinophilia; Purpura, Thrombocytopenic, Idiopathic; Rhinitis, Allergic, Seasonal; Sarcoidosis; Serum Sickness; Spondylitis, Ankylosing; Stevens-Johnson Syndrome; Synovitis; Tennis Elbow; Tenosynovitis; Thrombocytopenia; Thyroiditis, Subacute; Transfusion Reaction; Trichinellosis; Tuberculosis, Meningeal; Tuberculosis, Pulmonary; Uveitis, Posterior
Glucocorticoid receptor agonist
Small molecule
Approved
OTHER
ORAL
Altitude Sickness; Essential Tremor; Uterine Cervical Neoplasms; Glaucoma; Glaucoma, Open-Angle
Carbonic anhydrase II inhibitor
Small molecule
Approved
Unknown
Unknown
Anemia, Diamond-Blackfan; Psychotic Disorders
Unknown
Small molecule
Approved
Unknown
Unknown
Glaucoma
Unknown
Small molecule
Approved
OTHER
INJECTION; ORAL; SUBCUTANEOUS
Pregnancy; Alzheimer Disease; Breast Neoplasms; HIV Infections; Pain; Primary Ovarian Insufficiency; Sleep Apnea Syndromes; Bone Diseases; Cardiovascular Diseases; Coronary Disease; Diabetes Mellitus; Endometrial Neoplasms; Heart Diseases; Hot Flashes; Hypercholesterolemia; Hypertension; Infertility; Kidney Neoplasms; Lupus Erythematosus, Systemic; Menopause; Menorrhagia; Myocardial Ischemia; Osteoporosis; Prostatic Neoplasms; Thrombosis; Turner Syndrome; Carcinoma, Renal Cell; Endometriosis; Hyperplasia; Neoplasms; Uterine Hemorrhage
Progesterone receptor agonist
Small molecule
Approved
OTHER
ORAL
Cardiovascular Diseases
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
OTHER
OPHTHALMIC
Unknown
Acetylcholinesterase inhibitor
Small molecule
Approved
Unknown
Unknown
Chronic Pain; Pain
Unknown
Small molecule
Approved
OTHER
ORAL
Cardiovascular Diseases
Thiazide-sensitive sodium-chloride cotransporter inhibitor
Small molecule
Approved
OTHER
ORAL
Alcoholism; Chorioretinitis; Diabetes Mellitus; Diabetic Nephropathies; Dry Eye Syndromes; Leukemia; Leukemia, Myeloid, Acute; Melanosis; Non-alcoholic Fatty Liver Disease; Arrhythmogenic Right Ventricular Dysplasia; Cardiomyopathies; Cerebral Hemorrhage; Fatty Liver; Hypertension, Pulmonary; Macular Degeneration; Neoplasms; Neuroblastoma; Polycystic Ovary Syndrome; Puberty, Precocious; Severe Acute Respiratory Syndrome; Acne Vulgaris; Acute Kidney Injury; Aortic Valve Stenosis; Arthritis, Rheumatoid; Atrial Fibrillation; Heart Failure, Diastolic; Muscular Dystrophy, Duchenne; Non-ST Elevated Myocardial Infarction; Polycystic Kidney, Autosomal Dominant; Renal Insufficiency, Chronic; ST Elevation Myocardial Infarction; Ascites; Cardiovascular Diseases; Edema; Essential Hypertension; Fibrosis; Heart Failure; Hyperaldosteronism; Hypertension; Liver Cirrhosis; Myocardial Infarction; Nephrotic Syndrome; Toxemia
Mineralocorticoid receptor antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Mu opioid receptor agonist
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Compartment Syndromes; Osteoarthritis, Hip; Osteoarthritis, Knee; Pain
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
OTHER
OPHTHALMIC
Ocular Hypertension; Parkinson Disease; Presbyopia; Sialorrhea; Eye Diseases; Mydriasis
Muscarinic acetylcholine receptor M3 antagonist