Display Options:
Total: 6532
Small molecule
Investigational
Unknown
Unknown
Low Back Pain; Arthritis, Rheumatoid; Back Pain; Dysmenorrhea; Rheumatic Diseases
Unknown
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
Small molecule
Investigational
Unknown
Unknown
Severe Acute Respiratory Syndrome; Venous Thrombosis; Multiple Myeloma; Leukemia, Myeloid, Acute
Selectin E antagonist
Small molecule
Investigational
Unknown
Unknown
Anxiety; Deglutition Disorders; Dementia; Depressive Disorder; Schizophrenia; Cardiovascular Diseases
Unknown
Small molecule
Investigational
Unknown
Unknown
Liver Diseases; Hyperuricemia; Gout
Solute carrier family 22 member 12 inhibitor
Small molecule
Investigational
Unknown
Unknown
Carcinoma, Non-Small-Cell Lung; Carcinoma, Transitional Cell; Lung Neoplasms; Penile Neoplasms; Prostatic Neoplasms, Castration-Resistant; Small Cell Lung Carcinoma; Stomach Neoplasms; Breast Neoplasms; Head and Neck Neoplasms; Neoplasms; Urinary Bladder Neoplasms; Urogenital Neoplasms
Tubulin inhibitor
Small molecule
Investigational
Unknown
Unknown
Hyperlipoproteinemias; Kidney Diseases; Liver Diseases; Constipation; Hepatitis C; Non-alcoholic Fatty Liver Disease
Diacylglycerol O-acyltransferase 1 inhibitor
Small molecule
Investigational
Unknown
Unknown
Varicose Veins
Unknown
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
Small molecule
Investigational
Unknown
Unknown
Glaucoma; Ocular Hypertension; Osteoarthritis, Knee; Severe Acute Respiratory Syndrome; Uveitis, Intermediate; Uveitis, Posterior; Arthritis, Rheumatoid; Dry Eye Syndromes; Psoriasis
Adenosine A3 receptor agonist
Small molecule
Investigational
Unknown
Unknown
Hyperlipidemias; Lipid Metabolism Disorders; Severe Acute Respiratory Syndrome; Acute Coronary Syndrome; Cardiovascular Diseases; Coronary Disease; Dyslipidemias; Peripheral Arterial Disease
Cholesteryl ester transfer protein inhibitor
Small molecule
Investigational
Unknown
Unknown
Breast Neoplasms; Neoplasms; Polycystic Kidney, Autosomal Recessive; Brain Neoplasms; Glioblastoma; Polycystic Kidney, Autosomal Dominant; Carcinoma, Non-Small-Cell Lung
Ephrin type-B receptor 4 inhibitor
Small molecule
Investigational
Unknown
Unknown
Astrocytoma; Brain Neoplasms; Carcinoma, Non-Small-Cell Lung; Glioblastoma; Glioma; Gliosarcoma; Leukemia, Biphenotypic, Acute; Leukemia, Erythroblastic, Acute; Leukemia, Megakaryoblastic, Acute; Leukemia, Monocytic, Acute; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Leukemia, Myelomonocytic, Acute; Leukemia, Promyelocytic, Acute; Myelodysplastic Syndromes; Neoplasms; Oligodendroglioma; Ovarian Neoplasms; Breast Neoplasms; Carcinoma, Renal Cell; Colonic Neoplasms; Gastrointestinal Stromal Tumors; Head and Neck Neoplasms; Kidney Neoplasms; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma; Melanoma; Pancreatic Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Waldenstrom Macroglobulinemia; Colorectal Neoplasms; Multiple Myeloma
Unknown
Small molecule
Investigational
Unknown
Unknown
Diabetic Neuropathies; Stroke
Unknown
Small molecule
Investigational
Unknown
Unknown
Cognitive Dysfunction; Schizophrenia; Alzheimer Disease
Serotonin 6 (5-HT6) receptor antagonist
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
Small molecule
Investigational
Unknown
Unknown
Astrocytoma; Carcinoma, Non-Small-Cell Lung; Colorectal Neoplasms; Glioblastoma; Oligodendroglioma; Ovarian Neoplasms; Breast Neoplasms; Neoplasms
DNA topoisomerase I inhibitor
Small molecule
Investigational
Unknown
Unknown
Angioedemas, Hereditary
Plasma kallikrein inhibitor
Small molecule
Investigational
Unknown
Unknown
Dry Eye Syndromes; Neuralgia, Postherpetic; Arthralgia; Myalgia; Osteoarthritis, Knee; Pain
Vanilloid receptor agonist
Small molecule
Investigational
Unknown
Unknown
Sleep Initiation and Maintenance Disorders
Orexin receptor antagonist
Small molecule
Investigational
Unknown
Unknown
Esophageal Neoplasms; Purpura, Thrombocytopenic, Idiopathic
Unknown
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
Small molecule
Investigational
Unknown
Unknown
Cystic Fibrosis
Cystic fibrosis transmembrane conductance regulator positive modulator
Small molecule
Investigational
Unknown
Unknown
Unknown
Unknown
Small molecule
Investigational
Unknown
Unknown
Parkinson Disease
Dopamine receptors; D2 & D3 partial agonist
Small molecule
Investigational
Unknown
Unknown
Carcinoma, Hepatocellular; Glioblastoma; Hematologic Neoplasms; Neoplasms; Squamous Cell Carcinoma of Head and Neck; Stomach Neoplasms; Urinary Bladder Neoplasms; Carcinoma, Non-Small-Cell Lung; Head and Neck Neoplasms; Lung Neoplasms; Melanoma; Skin Neoplasms
Indoleamine 2,3-dioxygenase inhibitor
Small molecule
Investigational
Unknown
Unknown
Diabetes Mellitus, Type 2; Pituitary ACTH Hypersecretion; Adrenal Gland Diseases; Adrenocortical Hyperfunction; Cushing Syndrome
Cytochrome P450 11A1 inhibitor
Small molecule
Investigational
Unknown
Unknown
Esophageal Neoplasms; Melanoma; Neoplasms; Lymphoma, Mantle-Cell; Ovarian Neoplasms; Myelodysplastic Syndromes
Cellular tumor antigen p53 stabiliser
Small molecule
Investigational
Unknown
Unknown
Osteoarthritis, Knee; Complex Regional Pain Syndromes
Unknown
Small molecule
Investigational
Unknown
Unknown
Cocaine-Related Disorders; Psychotic Disorders; Schizophrenia
Unknown
Small molecule
Investigational
Unknown
Unknown
Osteomyelitis; Bacterial Infections
Bacterial 70S ribosome inhibitor
Small molecule
Investigational
Unknown
Unknown
Carcinoma, Renal Cell; Urinary Bladder Neoplasms; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant
Unknown
Small molecule
Investigational
Unknown
Unknown
Liver Diseases; Duodenal Ulcer; Gastroesophageal Reflux; Helicobacter Infections; Laryngopharyngeal Reflux; Peptic Ulcer; Stomach Ulcer
Potassium-transporting ATPase blocker
Small molecule
Investigational
Unknown
Unknown
Liver Diseases; Neoplasms; Diabetes Mellitus; Diabetes Mellitus, Type 2; Kidney Diseases
Dipeptidyl peptidase IV inhibitor
Small molecule
Investigational
Unknown
Unknown
Osteomyelitis; Eye Infections; Nasal Obstruction
Unknown